SCHEMBL7862960

SCHEMBL7862960

Bc1c(-c2cccc3ccccc23)noc1[C@H]1CNCC[C@H]1O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.42
REN P00797 1/20 0.42
GABRA1 P14867 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
HTR2A P28223 2/20 0.38
DRD2 P14416 1/20 0.37
HRH3 Q9Y5N1 1/20 0.34
ESR1 P03372 2/20 0.34
ESR2 Q92731 2/20 0.34
PRKD3 O94806 1/20 0.34
PRKD1 Q15139 1/20 0.34
PRKD2 Q9BZL6 1/20 0.34
CCNK O75909 1/20 0.32
CDK7 P50613 1/20 0.32
CCNH P51946 1/20 0.32
MNAT1 P51948 1/20 0.32
CDK12 Q9NYV4 1/20 0.32
NISCH Q9Y2I1 1/20 0.32
BCHE P06276 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7874302 0.71 REN (0.52) KCNH2RENGABRA1GABRG2GABRB3
SCHEMBL6042859 0.63 KDM1A (0.47) HTR2A
SCHEMBL10964208 0.61 SLC18A3 (0.54) HTR2ADRD2MAPT
SCHEMBL5923778 0.61 SLC18A3 (0.54) HTR2ADRD2MAPT
SCHEMBL10964458 0.61 SLC18A3 (0.54) HTR2ADRD2MAPT
SCHEMBL10964453 0.61 SLC18A3 (0.54) HTR2ADRD2MAPT
SCHEMBL8273744 0.61 SLC18A3 (0.54) HTR2ADRD2MAPT
Hydrochloric Acid SCHEMBL193499 0.59 NR1H4 (0.44) KDM4EALDH1A1TP53MAPTHPGD
SCHEMBL18790802 0.57 GRIN2D (0.40) HTR2AKDM4EALDH1A1MAPTHPGD
SCHEMBL11242027 0.57 SLC6A2 (0.45) HTR2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed