SCHEMBL7863682

SCHEMBL7863682

Cc1ccnc(-c2nccc(C)c2C(=O)O)c1.[Ru].c1ccc(-c2ccnc(-c3cc(-c4ccccc4)ccn3)c2)cc1.c1ccc(-c2ccnc(-c3cc(-c4ccccc4)ccn3)c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.44
CYP2A6 P11509 1/20 0.42
CCR1 P32246 1/20 0.41
CCR5 P51681 1/20 0.41
CCR8 P51685 1/20 0.41
DHODH Q02127 2/20 0.40
KMO O15229 1/20 0.40
MEN1 O00255 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
GRM5 P41594 1/20 0.38
KDM4C Q9H3R0 3/20 0.38
KDM4A O75164 2/20 0.38
KDM2B Q8NHM5 1/20 0.37
LDHA P00338 1/20 0.37
EGFR P00533 1/20 0.37
SMO Q99835 2/20 0.37
WNT3A P56704 1/20 0.37
CNR1 P21554 1/20 0.37
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30447581 0.87 CCR1 (0.50) PDE10ACYP2A6CCR1CCR5CCR8
SCHEMBL14224575 0.80 CCR1 (0.65) CYP2A6CCR1CCR5CCR8MEN1
SCHEMBL30447562 0.80 CCR1 (0.42) PDE10ACYP2A6CCR1CCR5CCR8
SCHEMBL5532401 0.77 DHODH (0.49) PDE10ADHODHMEN1KMT2ALDHA
SCHEMBL645855 0.76 KDM4E (0.49) CCR1CCR5CCR8DHODHKMT2A
SCHEMBL30447796 0.73 CCR1 (0.47) PDE10ACYP2A6CCR1CCR5CCR8
SCHEMBL3235044 0.72 CCR1 (0.74) CYP2A6CCR1CCR5CCR8MEN1
SCHEMBL2789829 0.72 ASIC3 (0.52) KDM4CKDM4AEGFRSMOCNR1
SCHEMBL7853202 0.71 CCR1 (0.61) CYP2A6CCR1CCR5CCR8KMO
SCHEMBL19009238 0.70 CYP2A6 (0.61) PDE10ACYP2A6CCR1CCR5CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20010018194-A1 Luminescence assays LJL BIOSYSTEMS, INC. 2001-08-30 US disclosed
WO-2000023785-A2 IMPROVEMENTS IN LUMINESCENCE ASSAYS LJL BIOSYSTEMS, INC. (US) 2000-04-27 WO disclosed