SCHEMBL7864155

SCHEMBL7864155

COC(=O)C1=C(c2ccc(-n3c(C)nc4cnccc43)cc2)NC(C)=C(C(=O)OC(C)C#Cc2cccnc2)C1CC(c1ccccc1)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 2/20 0.33
ITGA4 P13612 2/20 0.33
ADORA3 P0DMS8 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8135155 0.86 ADORA3 (0.40) ADORA3
SCHEMBL7873273 0.85 ADORA3 (0.39) ADORA3MEN1KMT2A
SCHEMBL7873331 0.83 MAPT (0.36) ADORA3MEN1KMT2A
SCHEMBL7864153 0.83 ADORA3 (0.39) ADORA3
SCHEMBL8138174 0.81 ADORA3 (0.36) ADORA3
SCHEMBL7864187 0.81 ADORA3 (0.39) ADORA3
SCHEMBL7876067 0.79 ADORA3 (0.38) ADORA3
SCHEMBL7876028 0.79 ADORA3 (0.38) ADORA3
SCHEMBL7869604 0.77 ADORA3 (0.40) ADORA3
SCHEMBL7864225 0.77 ADORA3 (0.41) ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306853-B1 DICARBOXYLIC ESTER DERIVATIVES OF DIHYDROPYRIDINE COMPOUNDS NIKKEN CHEMICALS CO., LTD. (JP) 2001-10-23 US disclosed