SCHEMBL7876028

SCHEMBL7876028

CCOC(=O)C1=C(c2cccc(-n3c(C)nc4cnccc43)c2)NC(C)=C(C(=O)OC(C)C#Cc2cccnc2)C1CCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 8/20 0.38
CACNA1C Q13936 2/20 0.35
TMIGD3 P0DMS9 1/20 0.35
TRPV1 Q8NER1 1/20 0.34
MAPK1 P28482 2/20 0.34
MAPT P10636 1/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
GRM5 P41594 1/20 0.33
ALDH1A1 P00352 2/20 0.32
LMNA P02545 1/20 0.32
ALOX12 P18054 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7873273 0.93 ADORA3 (0.39) ADORA3TMIGD3TRPV1MAPK1MAPT
SCHEMBL8144758 0.90 ADORA3 (0.39) ADORA3CACNA1CTMIGD3TRPV1MAPK1
SCHEMBL7876031 0.89 ADORA3 (0.39) ADORA3CACNA1CTMIGD3TRPV1MAPK1
SCHEMBL7873331 0.85 MAPT (0.36) ADORA3TMIGD3TRPV1MAPK1MAPT
SCHEMBL7873283 0.83 ADORA3 (0.40) ADORA3TMIGD3TRPV1MAPK1CYP3A4
SCHEMBL7864221 0.82 ADORA3 (0.40) ADORA3TMIGD3TRPV1MAPK1MAPT
SCHEMBL7876067 0.82 ADORA3 (0.38) ADORA3CACNA1CTMIGD3TRPV1MAPK1
SCHEMBL7864247 0.81 ADORA3 (0.34) ADORA3MAPK1MAPT
SCHEMBL7873247 0.81 ADORA3 (0.41) ADORA3CACNA1CTMIGD3TRPV1MAPK1
SCHEMBL8143535 0.80 ADORA3 (0.40) ADORA3TMIGD3TRPV1MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306853-B1 DICARBOXYLIC ESTER DERIVATIVES OF DIHYDROPYRIDINE COMPOUNDS NIKKEN CHEMICALS CO., LTD. (JP) 2001-10-23 US disclosed
EP-1055672-A1 1,4-DIHYDROPYRIDINE DERIVATIVES Nikken Chemicals Company, Limited (JP) 2000-11-29 EP disclosed