SCHEMBL7864166

SCHEMBL7864166

COC(=O)CC(=O)c1cccc(-n2ccnc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.52
PDE4A P27815 1/20 0.52
PDE4B Q07343 1/20 0.52
PDE4C Q08493 1/20 0.52
PDE4D Q08499 1/20 0.52
ABL1 P00519 1/20 0.52
IDO1 P14902 1/20 0.50
CYP3A4 P08684 2/20 0.46
BAZ2B Q9UIF8 1/20 0.46
CYP4Z1 Q86W10 1/20 0.46
MAPT P10636 2/20 0.44
PLOD2 O00469 1/20 0.44
PLOD3 O60568 1/20 0.44
PLOD1 Q02809 1/20 0.44
LMNA P02545 1/20 0.44
ROCK2 O75116 1/20 0.43
HDAC1 Q13547 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7869625 0.89 PDE4A (0.52) HTTPDE4APDE4BPDE4CPDE4D
SCHEMBL5868879 0.88 L3MBTL1 (0.51) HTTPDE4APDE4BPDE4CPDE4D
SCHEMBL5868816 0.85 IDO1 (0.54) HTTPDE4APDE4BPDE4CPDE4D
SCHEMBL7289319 0.84 HTT (0.69) HTTPDE4APDE4BPDE4CPDE4D
SCHEMBL5868840 0.84 HTT (0.69) HTTPDE4APDE4BPDE4CPDE4D
SCHEMBL10851507 0.84 PDE4A (0.59) HTTPDE4APDE4BPDE4CPDE4D
SCHEMBL7280094 0.79 CYP3A4 (0.67) HTTPDE4APDE4BPDE4CPDE4D
SCHEMBL10663235 0.79 IDO1 (0.52) PDE4APDE4BPDE4CPDE4DABL1
SCHEMBL4081415 0.78 L3MBTL1 (0.58) HTTPDE4APDE4BPDE4CPDE4D
SCHEMBL19031379 0.78 IDO1 (0.51) HTTPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306853-B1 DICARBOXYLIC ESTER DERIVATIVES OF DIHYDROPYRIDINE COMPOUNDS NIKKEN CHEMICALS CO., LTD. (JP) 2001-10-23 US disclosed
EP-1055672-A1 1,4-DIHYDROPYRIDINE DERIVATIVES Nikken Chemicals Company, Limited (JP) 2000-11-29 EP disclosed
US-4734415-A CARDIOTONIC, HYPOTENSIVE WARNER-LAMBERT COMPANY (US) 1988-03-29 US disclosed