SCHEMBL7865623

SCHEMBL7865623

O=C(Nc1ccccc1Br)Nc1ccc(Br)c2[nH]c(C(F)(F)F)nc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.47
CXCR2 P25025 10/20 0.46
ADRB3 P13945 1/20 0.46
TSPO P30536 1/20 0.46
SLC6A3 Q01959 1/20 0.46
TRPV1 Q8NER1 1/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
NPC1 O15118 1/20 0.45
LMNA P02545 1/20 0.45
RAB9A P51151 1/20 0.45
CXCR1 P25024 9/20 0.43
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
CASP3 P42574 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6816721 1.00 HTT (0.47) HTTCXCR2ADRB3TSPOSLC6A3
SCHEMBL7865622 0.91 HTT (0.47) HTTCXCR2ADRB3TSPOSLC6A3
SCHEMBL6817174 0.87 CXCR2 (0.60) HTTCXCR2ADRB3TSPOSLC6A3
SCHEMBL6817172 0.82 CXCR2 (0.60) HTTCXCR2ADRB3TSPOSLC6A3
SCHEMBL29116821 0.73 CSNK2A1 (0.56) MEN1KMT2AGAAMAPTTDP1
SCHEMBL30669533 0.73 CSNK2A1 (0.56) MEN1KMT2AGAAMAPTTDP1
SCHEMBL13235126 0.71 HTT (0.81) HTTCXCR2MEN1KMT2ANPC1
SCHEMBL27576138 0.70 PARP1 (0.40) MEN1KMT2AGAAMAPTTDP1
SCHEMBL6816893 0.68 MAPT (0.51) MEN1KMT2AGAAMAPTCASP3
SCHEMBL5595017 0.67 CXCR1 (0.68) HTTCXCR2MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6300325-B1 HETEROCYCLIC RECEPTOR ANTAGONIST SMITHKLINE BEECHAM CORPORATION 2001-10-09 US disclosed