SCHEMBL7865743

SCHEMBL7865743

NCc1ccc2c(c1)C(N)CC2

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 9/20 0.43
HTR1A P08908 1/20 0.41
DRD2 P14416 1/20 0.41
HTR2A P28223 1/20 0.41
KCNH2 Q12809 1/20 0.41
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39
HTR6 P50406 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7875148 0.98 ACHE (0.45) ACHEHTR1ADRD2HTR2AKCNH2
SCHEMBL21065657 0.84 ACHE (0.48) ACHEHTR1ADRD2HTR2AKCNH2
SCHEMBL8781041 0.82 ACHE (0.43) ACHEHTR1ADRD2HTR2AKCNH2
SCHEMBL27827581 0.80 ACHE (0.42) ACHEHTR1ADRD2HTR2AKCNH2
SCHEMBL19978162 0.80 HTR1A (0.43) ACHEHTR1ADRD2HTR2AKCNH2
SCHEMBL7369494 0.78 ACHE (0.39) ACHEHTR1ADRD2HTR2AKCNH2
SCHEMBL1004804 0.75 HTR2C (0.47) ACHEHTR1AHTR2AKCNH2
SCHEMBL7895243 0.75 HTR2C (0.47) ACHEHTR1AHTR2AKCNH2
SCHEMBL2038159 0.75 ACHE (0.45) ACHEHTR6
SCHEMBL30918006 0.75 ACHE (0.45) ACHEHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37438-E1 Acetamidine derivatives and their use as inhibitors for the nitric oxide synthase GLAXO WELLCOME INC. 2001-11-06 US disclosed
US-5866612-A Acetamidine derivatives and their use as inhibitors for the nitric oxide synthase GLAXO WELLCOME INC. (US) 1999-02-02 US disclosed
EP-0799191-A1 ACETAMIDINE DERIVATIVES AND THEIR USE AS INHIBITORS FOR THE NITRIC OXIDE SYNTHASE THE WELLCOME FOUNDATION LIMITED (GB) 1997-10-08 EP disclosed
WO-1996019440-A1 ACETAMIDINE DERIVATIVES AND THEIR USE AS INHIBITORS FOR THE NITRIC OXIDE SYNTHASE THE WELLCOME FOUNDATION LIMITED (GB) 1996-06-27 WO disclosed