SCHEMBL7877658

SCHEMBL7877658

CN/C=C(\C=N)c1cnc2[nH]cc(C(=O)c3cc(NS(=O)(=O)c4cccc(OC(F)(F)F)c4)ccc3F)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.42
KIT P10721 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
CYP2C9 P11712 3/20 0.39
CCR9 P51686 1/20 0.37
PIK3CA P42336 1/20 0.36
CYP2D6 P10635 1/20 0.36
BRAF P15056 1/20 0.36
SLC40A1 Q9NP59 1/20 0.36
NAMPT P43490 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7869062 0.89 CYP3A4 (0.44) CYP3A4KITHDAC1HDAC8CYP2C9
SCHEMBL7880231 0.89 CYP3A4 (0.53) CYP3A4KITHDAC3HDAC4HDAC1
SCHEMBL7869096 0.88 CYP3A4 (0.45) CYP3A4KITCYP2C9PIK3CABRAF
SCHEMBL298324 0.85 CYP3A4 (0.47) CYP3A4KITHDAC3HDAC4HDAC1
SCHEMBL298424 0.82 SLC40A1 (0.48) CYP3A4KITHDAC3HDAC4HDAC1
SCHEMBL7868957 0.81 CYP3A4 (0.51) CYP3A4CYP2C9PIK3CA
SCHEMBL298752 0.80 PAK1 (0.44) CYP3A4KITHDAC3HDAC4HDAC1
SCHEMBL12703796 0.80 CYP3A4 (0.59) CYP3A4KITCYP2C9CYP2D6BRAF
SCHEMBL7872497 0.79 BRAF (0.56) CYP3A4KITCYP2C9CYP2D6BRAF
SCHEMBL7876631 0.79 BRAF (0.38) CYP3A4KITCYP2C9BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010129570-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS PLEXXIKON, INC. (US) 2010-11-11 WO disclosed