SCHEMBL7869745

SCHEMBL7869745

Cc1sccc1C=CC(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 3/20 0.47
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA4 P22748 2/20 0.44
NFKB1 P19838 1/20 0.44
MIF P14174 1/20 0.43
HDAC3 O15379 1/20 0.41
TNKS O95271 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
TNKS2 Q9H2K2 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
ALDH1A1 P00352 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28748955 0.82 ALDH1A1 (0.41) HCAR2CA1CA2CA4NFKB1
SCHEMBL6296284 0.80 ALDH1A1 (0.38) ALDH1A1SMN1; SMN2NPC1RAB9AMAPK1
SCHEMBL6296286 0.80 ALDH1A1 (0.38) ALDH1A1SMN1; SMN2NPC1RAB9AMAPK1
SCHEMBL12078966 0.78 CA1 (0.50) HCAR2CA1CA2CA4NFKB1
SCHEMBL9756876 0.77 HCAR2 (0.47) HCAR2CA1CA2CA4NFKB1
SCHEMBL9756874 0.77 HCAR2 (0.47) HCAR2CA1CA2CA4NFKB1
SCHEMBL13245829 0.77 ALDH1A1 (0.37) ALDH1A1SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL7776471 0.74 RARA (0.48) HDAC1ALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL5283644 0.73 HCAR2 (0.47) HCAR2HDAC3TNKSHDAC4HDAC1
SCHEMBL5283646 0.73 HCAR2 (0.47) HCAR2HDAC3TNKSHDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100381566-C Recombinant methods and materials for producing epothilone and derivatives thereof KOSAN BIOSCIENCES INC (US) 2008-04-16 CN disclosed
CN-1333820-A Recombinant methods and materials for producing epothilone and eopthilone derivatives KOSAN BIOSCIENCES INC (US) 2002-01-30 CN disclosed
US-6303593-B1 FOR THERAPY HUMAN IMMUNODEFICIENCY VIRUS INFECTION, AQUIRED IMMUNODEFICIENCY SYNDROME (AIDS), INFLAMMATORY AND IMMUNOREGULATORY DISORDER OR DISEASE, ASTHMA, ALLERGIC RHINITIS, DERMATITIS, CONJUNCTIVITIS, ATHEROSCLEROSIS MERCK & CO., INC. 2001-10-16 US disclosed
WO-2000051608-A1 3-THIENYL AND 3-FURANYL PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-09-08 WO disclosed