SCHEMBL7870941

SCHEMBL7870941

COC(=O)C(C(C)c1ccc(N)cc1)C1CCCN1C

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 2/20 0.46
CHRNB4 P30926 4/20 0.40
CHRNA3 P32297 4/20 0.40
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14193555 0.89 CHRNB4 (0.41) CHRNB4CHRNA3
SCHEMBL31575359 0.78 CHRNB2 (0.43) SLC6A3CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL31575321 0.78 DPP4 (0.46) CHRNB4CHRNA3
SCHEMBL31575334 0.78 DPP4 (0.46) CHRNB4CHRNA3
SCHEMBL31575348 0.78 CHRNB2 (0.43) SLC6A3CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL31575342 0.74 DPP4 (0.45) SLC6A3
SCHEMBL31575328 0.74 SLC6A2 (0.44) SLC6A3CHRNB2CHRNA4
SCHEMBL30166180 0.74 SLC6A2 (0.44) SLC6A3CHRNB2CHRNA4
SCHEMBL10082491 0.71 CHRNA7 (0.50) CHRNB4CHRNA3CHRNB2CHRNA4
SCHEMBL23886115 0.71 CHRNB4 (0.42) CHRNB4CHRNA3CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316490-B1 FOR THERAPY OF PARKINSON'S DISEASE, ALZHEIMER'S DISEASE, DEMENTIA, CONTROLLING PAIN MERCK & CO., INC. 2001-11-13 US disclosed
EP-0874818-A1 NOVEL SUBSTITUTED ARYL COMPOUNDS USEFUL AS MODULATORS OF ACETYLCHOLINE RECEPTORS SIBIA NEUROSCIENCES, INC. (US) 1998-11-04 EP disclosed
WO-1997019059-A1 NOVEL SUBSTITUTED ARYL COMPOUNDS USEFUL AS MODULATORS OF ACETYLCHOLINE RECEPTORS SIBIA NEUROSCIENCES, INC. (US) 1997-05-29 WO disclosed