SCHEMBL7871830

SCHEMBL7871830

NC(=O)c1c(C(=O)O)[nH]c2cc(O)c(O)cc12

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 12/20 0.60
SRC P12931 4/20 0.45
PRKACA P17612 3/20 0.45
PRKACG P22612 3/20 0.45
PRKACB P22694 3/20 0.45
APP P05067 1/20 0.36
MAP2 P11137 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27948924 0.87 GPR35 (0.66) GPR35SRCPRKACAPRKACGPRKACB
SCHEMBL9425166 0.79 GPR35 (0.60) GPR35SRCPRKACAPRKACGPRKACB
SCHEMBL1155981 0.77 NGFR (0.53) MAP2
SCHEMBL11784003 0.77 GPR35 (0.66) GPR35SRCPRKACAPRKACGPRKACB
SCHEMBL27442503 0.76 MAP2 (0.59) MAP2
SCHEMBL1156019 0.75 CA1 (0.62)
SCHEMBL14703001 0.75 GPR35 (0.64) GPR35SRCPRKACAPRKACGPRKACB
SCHEMBL721793 0.74 MAP2 (0.58) MAP2
SCHEMBL31120728 0.71 PRNP (0.61) GPR35SRCPRKACAPRKACGPRKACB
SCHEMBL1156584 0.71 POLB (0.68)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6313313-B1 WATER SOLUBLE CATIONIC AMIDE OR ESTER MADE FROM REACTION WITH 5,6-DIHYDROXYINDOLE-2-CARBOXYLIC ACID BRISTOL-MYERS SQUIBB COMPANY 2001-11-06 US disclosed
EP-0865269-A4 SYNTHESIS OF QUATERNARY MELANIN COMPOUNDS AND THEIR USE AS HAIR DYES OR FOR SKIN TREATMENT BRISTOL MYERS SQUIBB CO (US) 2000-01-19 EP disclosed
US-5827330-A OXIDATIVE POLYMERIZATION OF 5,6-DIHYDROXYINDOLE QUATERNARY AMINE DERIVATIVES BRISTOL-MYERS SQUIBB CO. (US) 1998-10-27 US disclosed
EP-0865269-A1 SYNTHESIS OF QUATERNARY MELANIN COMPOUNDS AND THEIR USE AS HAIR DYES OR FOR SKIN TREATMENT Bristol-Myers Squibb Company (US) 1998-09-23 EP disclosed
US-5702712-A Melanoquaternary compounds and their use as hair dyes and for skin treatment CLAIROL, INCORPORATED (US) 1997-12-30 US disclosed
US-5686084-A Synthesis of quaternary melanin compounds and their use as hair dyes or for skin treatment CLAIROL INCORPORATED (US) 1997-11-11 US disclosed
WO-1997020542-A1 SYNTHESIS OF QUATERNARY MELANIN COMPOUNDS AND THEIR USE AS HAIR DYES OR FOR SKIN TREATMENT BRISTOL-MYERS SQUIBB COMPANY (US) 1997-06-12 WO disclosed