SCHEMBL7873253

SCHEMBL7873253

CCOC(=O)C1=C(c2ccc(-n3c(C)nc4cnccc43)cc2)NC(C)=C(C(=O)OCC#Cc2cccnc2)C1/C=C/c1ccccc1OC

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.48
KDM4E B2RXH2 3/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
ALDH1A1 P00352 2/20 0.48
LMNA P02545 1/20 0.48
HTT P42858 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
ADORA3 P0DMS8 10/20 0.43
TMIGD3 P0DMS9 2/20 0.40
TSHR P16473 2/20 0.35
USP2 O75604 1/20 0.35
HPGD P15428 1/20 0.34
XBP1 P17861 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7869556 0.93 ADORA3 (0.43) MAPTKDM4EMEN1KMT2AALDH1A1
SCHEMBL7876063 0.91 ADORA3 (0.52) MAPTKDM4EMEN1KMT2AALDH1A1
SCHEMBL7864190 0.88 ADORA3 (0.43) MAPTKDM4EMEN1KMT2AALDH1A1
SCHEMBL8136874 0.88 ADORA3 (0.40) ALDH1A1ADORA3TMIGD3TSHRHPGD
SCHEMBL7872534 0.86 ADORA3 (0.38) MAPTADORA3TMIGD3TSHR
SCHEMBL7873370 0.86 ADORA3 (0.37) ADORA3TMIGD3TSHR
SCHEMBL7872512 0.86 ADORA3 (0.38) ADORA3TMIGD3TSHR
SCHEMBL7871436 0.85 TSHR (0.38) ADORA3TMIGD3TSHR
SCHEMBL7864225 0.82 ADORA3 (0.41) ADORA3TMIGD3TSHR
SCHEMBL7872515 0.82 ADORA3 (0.38) MAPTADORA3TMIGD3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306853-B1 DICARBOXYLIC ESTER DERIVATIVES OF DIHYDROPYRIDINE COMPOUNDS NIKKEN CHEMICALS CO., LTD. (JP) 2001-10-23 US disclosed
EP-1055672-A1 1,4-DIHYDROPYRIDINE DERIVATIVES Nikken Chemicals Company, Limited (JP) 2000-11-29 EP disclosed