SCHEMBL7873370

SCHEMBL7873370

CCOC(=O)C1=C(c2ccc(-n3c(C)nc4cnccc43)cc2)NC(C)=C(C(=O)OCC#Cc2cccnc2)C1/C=C/C1CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.37
TMIGD3 P0DMS9 1/20 0.37
ITGB1 P05556 1/20 0.34
ITGA4 P13612 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7876063 0.89 ADORA3 (0.52) ADORA3TMIGD3
SCHEMBL7864205 0.89 TSHR (0.35) ADORA3TSHR
SCHEMBL8136874 0.87 ADORA3 (0.40) ADORA3TMIGD3TSHR
SCHEMBL7869556 0.87 ADORA3 (0.43) ADORA3TMIGD3TSHR
SCHEMBL7871436 0.87 TSHR (0.38) ADORA3TMIGD3TSHR
SCHEMBL7872512 0.86 ADORA3 (0.38) ADORA3TMIGD3TSHR
SCHEMBL7873253 0.86 MAPT (0.48) ADORA3TMIGD3TSHR
SCHEMBL7864163 0.86 ADORA3 (0.34) ADORA3TSHR
SCHEMBL7872515 0.84 ADORA3 (0.38) ADORA3TMIGD3TSHR
SCHEMBL7871376 0.83 ADORA3 (0.37) ADORA3TMIGD3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306853-B1 DICARBOXYLIC ESTER DERIVATIVES OF DIHYDROPYRIDINE COMPOUNDS NIKKEN CHEMICALS CO., LTD. (JP) 2001-10-23 US disclosed
EP-1055672-A1 1,4-DIHYDROPYRIDINE DERIVATIVES Nikken Chemicals Company, Limited (JP) 2000-11-29 EP disclosed