SCHEMBL7873339

SCHEMBL7873339

CC[C@H](C)CC(=O)N(C[C@H](C)Cc1cccc(N(CC(C)C)S(=O)(=O)c2ccccc2)c1O)NC(=O)CNC1CC1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 4/20 0.34
BCL2L1 Q07817 3/20 0.34
KDM4E B2RXH2 3/20 0.33
MAPT P10636 1/20 0.33
RORC P51449 7/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7584650 0.85 KMT2A (0.37) MCL1BCL2L1KDM4ERORCALDH1A1
SCHEMBL7584634 0.80 NPC1 (0.39) MCL1BCL2L1KDM4ERORCALDH1A1
SCHEMBL6392313 0.79 KEAP1 (0.37) MAPTRORCALDH1A1MEN1KMT2A
SCHEMBL6387295 0.75 RORC (0.33) MCL1BCL2L1RORCALDH1A1
SCHEMBL7584054 0.75 KMT2A (0.39) MCL1BCL2L1KDM4ERORCALDH1A1
SCHEMBL7876543 0.74 KEAP1 (0.39) MAPTRORCALDH1A1MEN1KMT2A
SCHEMBL6395395 0.74 KEAP1 (0.36) MCL1MAPTALDH1A1MEN1KMT2A
SCHEMBL7450756 0.73 CYP2C8 (0.33) MCL1BCL2L1MAPT
SCHEMBL7587276 0.73 KMT2A (0.37) MCL1BCL2L1KDM4ERORCALDH1A1
SCHEMBL7458622 0.72 RORC (0.45) MCL1BCL2L1RORCALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316496-B1 FOR THERAPY OF RETROVIRAL INFECTION; PROPHYLAXIS OF REPLICATION OF RETROVIRUS, THERAPY OF AIDS (ACQUIRED IMMUNE DEFICIENCY SYNDROME) G. D. SEARLE & CO. 2001-11-13 US disclosed