SCHEMBL7873436

SCHEMBL7873436

CC(C)(C)[C@H](N)C(=O)Nc1cnccc1N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CIT O14578 1/20 0.42
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
HDAC1 Q13547 5/20 0.38
HDAC3 O15379 3/20 0.38
HDAC2 Q92769 3/20 0.38
HDAC8 Q9BY41 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
KDM4C Q9H3R0 4/20 0.36
KDM6B O15054 2/20 0.36
MEN1 O00255 1/20 0.36
KDM4A O75164 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
KMT2A Q03164 1/20 0.36
KDM4D Q6B0I6 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15432245 0.83 XIAP (0.45) CITKDM4EALDH1A1GLAGAA
SCHEMBL6625479 0.76 CIT (0.52) CITKDM4ETDP1L3MBTL1
SCHEMBL7425368 0.76 CIT (0.52) CITKDM4ETDP1L3MBTL1
SCHEMBL14357917 0.76 HDAC1 (0.46) KDM4EALDH1A1GLAGAAHDAC1
SCHEMBL7868098 0.76 FFAR2 (0.56) KMT2AAHR
SCHEMBL28390904 0.75 NAMPT (0.47) KDM4EALDH1A1GLAGAA
Hydrochloric Acid SCHEMBL7868142 0.75 FFAR2 (0.54) KMT2AAHR
Hydrochloric Acid SCHEMBL7874804 0.75 FFAR2 (0.54) KMT2AAHR
Hydrochloric Acid SCHEMBL29373586 0.74 HDAC1 (0.45) KDM4EALDH1A1GLAGAAHDAC1
Hydrochloric Acid SCHEMBL5749683 0.74 HDAC1 (0.45) KDM4EALDH1A1GLAGAAHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6329400-B1 INHIBITION OR ANTAGONISM OF MATRIX METALLOPROTEASES, AND/OR TUMOR NECROSIS FACTOR-ALPHA; EXTRACELLULAR MATRIX DEGRADATION, INHIBITION OF SHEDDING OF CELL SURFACE PROTEIN ECTODOMAINS AND CD23 PROTEOLYSIS GLAXO WELLCOME INC. 2001-12-11 US disclosed