SCHEMBL7873697

SCHEMBL7873697

Cc1onc(-c2ccccn2)c1COc1cc(C(=O)NC(C)CO)nn1C

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 16/20 0.54
ITGA5 P08648 2/20 0.46
NTRK1 P04629 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2628078 1.00 GABRA5 (0.54) GABRA5ITGA5NTRK1
SCHEMBL298033 1.00 GABRA5 (0.54) GABRA5ITGA5NTRK1
SCHEMBL296603 0.93 GABRA5 (0.62) GABRA5ITGA5
SCHEMBL296088 0.87 GABRA5 (0.53) GABRA5NTRK1
SCHEMBL2628079 0.87 GABRA5 (0.53) GABRA5NTRK1
SCHEMBL296703 0.85 GABRA5 (0.60) GABRA5ITGA5
SCHEMBL2628069 0.85 GABRA5 (0.59) GABRA5ITGA5
SCHEMBL286341 0.85 GABRA5 (0.59) GABRA5ITGA5
SCHEMBL7870299 0.85 GABRA5 (0.59) GABRA5ITGA5
SCHEMBL297966 0.85 GABRA5 (0.59) GABRA5ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127975-A1 ISOXAZOLE-PYRAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-11-11 WO disclosed