SCHEMBL7874771

SCHEMBL7874771

CCOC(=O)C(OC=O)[C@H]1CC[C@@H](c2cc(N(COCC[Si](C)(C)C)COCC[Si](C)(C)C)n3ncc(-c4ccc(-c5ccccc5)nc4)c3n2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 8/20 0.41
MTOR P42345 3/20 0.36
RPTOR Q8N122 3/20 0.36
MLST8 Q9BVC4 3/20 0.36
KDM4E B2RXH2 4/20 0.35
HSD17B10 Q99714 3/20 0.35
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
GPR119 Q8TDV5 3/20 0.33
NFKB1 P19838 2/20 0.33
NFKB2 Q00653 2/20 0.33
RELA Q04206 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
TP53 P04637 1/20 0.33
STAT1 P42224 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAPT P10636 1/20 0.32
CHEK1 O14757 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10237541 0.92 DGAT1 (0.40) DGAT1MTORRPTORMLST8KDM4E
SCHEMBL7875234 0.90 DGAT1 (0.42) DGAT1MTORRPTORMLST8KDM4E
SCHEMBL1024356 0.88 DGAT1 (0.52) DGAT1MTORRPTORMLST8KDM4E
SCHEMBL2680922 0.86 DGAT1 (0.40) DGAT1MTORRPTORMLST8KDM4E
SCHEMBL2680917 0.86 DGAT1 (0.40) DGAT1MTORRPTORMLST8KDM4E
SCHEMBL2680071 0.86 DGAT1 (0.41) DGAT1MTORRPTORMLST8KDM4E
SCHEMBL2680067 0.86 DGAT1 (0.41) DGAT1MTORRPTORMLST8KDM4E
SCHEMBL2723620 0.85 DGAT1 (0.43) DGAT1MTORRPTORMLST8HSD17B10
SCHEMBL7881214 0.85 DGAT1 (0.39) DGAT1MTORRPTORMLST8KDM4E
SCHEMBL2679692 0.84 DGAT1 (0.39) DGAT1MTORRPTORMLST8KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118207-A1 PYRAZOLO [1, 5-A] PYRIMIDINE DERIVATIVES AS MTOR INHIBITORS SCHERING CORPORATION (US) 2010-10-14 WO disclosed