SCHEMBL7875339

SCHEMBL7875339

O=C(O)C(=S)CC(=O)c1ccc(F)c(F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.50
CES1 P23141 2/20 0.50
ERCC5 P28715 2/20 0.40
FEN1 P39748 2/20 0.40
CHRNA1 P02708 1/20 0.40
CHRNG P07510 1/20 0.40
CHRNB1 P11230 1/20 0.40
CHRNB2 P17787 1/20 0.40
SLC6A2 P23975 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40
SLC6A3 Q01959 1/20 0.40
CHRND Q07001 1/20 0.40
ALDH1A1 P00352 2/20 0.39
DPP4 P27487 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
VNN1 O95497 1/20 0.39
MAOA P21397 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2582326 0.82 CES1 (0.57) CES2CES1ERCC5FEN1CHRNA1
SCHEMBL23709229 0.77 CES2 (0.55) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL7868669 0.76 TSHR (0.53)
SCHEMBL28771713 0.74 CES2 (0.57) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL1925141 0.74 PLOD2 (0.66) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL20491395 0.74 CES2 (0.52) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL25193546 0.74 MEN1 (0.54) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL2273688 0.74 CES2 (0.61) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL5253742 0.74 CES2 (0.61) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL671907 0.74 CES2 (0.61) CES2CES1CHRNA1CHRNGCHRNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6323240-B1 HALOGENATED DERIVATIVES AS ENZYME INHIBITORS PHARMACIA & UPJOHN S.P.A. (IT) 2001-11-27 US disclosed