SCHEMBL7876072

SCHEMBL7876072

CCOC(=O)C1=C(c2ccc(-n3c(C(C)C)nc4cnccc43)cc2)NC(C)=C(C(=O)OCC#Cc2cccnc2)C1CCc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 10/20 0.39
TMIGD3 P0DMS9 1/20 0.36
TRPV1 Q8NER1 2/20 0.36
MAPK1 P28482 2/20 0.36
MAPT P10636 1/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.35
GAA P10253 1/20 0.35
CACNA1C Q13936 2/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7871349 0.94 ADORA3 (0.38) ADORA3TMIGD3TRPV1MAPK1MAPT
SCHEMBL7873283 0.93 ADORA3 (0.40) ADORA3TMIGD3TRPV1MAPK1CYP3A4
SCHEMBL7864187 0.91 ADORA3 (0.39) ADORA3TMIGD3TRPV1MAPK1MAPT
SCHEMBL8135837 0.90 ADORA3 (0.34) ADORA3MAPK1MAPTCYP3A4TSHR
SCHEMBL8143535 0.89 ADORA3 (0.40) ADORA3TMIGD3TRPV1MAPK1MAPT
SCHEMBL7869551 0.88 ADORA3 (0.39) ADORA3TMIGD3TRPV1MAPK1MAPT
SCHEMBL8142233 0.88 CACNA1C (0.39) ADORA3TMIGD3MAPK1CYP3A4TSHR
SCHEMBL7864221 0.87 ADORA3 (0.40) ADORA3TMIGD3TRPV1MAPK1MAPT
SCHEMBL7864225 0.86 ADORA3 (0.41) ADORA3TMIGD3MAPK1CYP3A4TSHR
SCHEMBL8144758 0.86 ADORA3 (0.39) ADORA3TMIGD3TRPV1MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306853-B1 DICARBOXYLIC ESTER DERIVATIVES OF DIHYDROPYRIDINE COMPOUNDS NIKKEN CHEMICALS CO., LTD. (JP) 2001-10-23 US disclosed
EP-1055672-A1 1,4-DIHYDROPYRIDINE DERIVATIVES Nikken Chemicals Company, Limited (JP) 2000-11-29 EP disclosed