SCHEMBL7876348

SCHEMBL7876348

COc1cc(-n2nc(C(F)(F)F)cc2-c2ccc(S(C)(=O)=O)cc2)ccc1Cl

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.65
PTGS1 P23219 8/20 0.65
CYP2C9 P11712 2/20 0.65
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
TSHR P16473 1/20 0.56
CYP2C19 P33261 1/20 0.56
THPO P40225 1/20 0.56
BLM P54132 1/20 0.56
PMP22 Q01453 1/20 0.56
HIF1A Q16665 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8069691 0.92 PTGS2 (0.65) PTGS2PTGS1CYP2C9
SCHEMBL7876594 0.88 PTGS2 (0.70) PTGS2PTGS1CYP2C9
SCHEMBL7876487 0.87 PTGS2 (0.65) PTGS2PTGS1CYP2C9
SCHEMBL6719190 0.87 PTGS2 (0.59) PTGS2PTGS1CYP2C9CYP1A2CYP3A4
SCHEMBL7874446 0.87 PTGS2 (0.52) PTGS2PTGS1CYP2C9
SCHEMBL6736285 0.87 PTGS2 (0.52) PTGS2PTGS1CYP2C9CYP1A2CYP3A4
SCHEMBL7874468 0.86 PTGS2 (0.70) PTGS2PTGS1CYP2C9
SCHEMBL7878995 0.86 PTGS2 (0.73) PTGS2PTGS1CYP2C9CYP3A4TSHR
SCHEMBL7874455 0.85 PTGS2 (0.67) PTGS2PTGS1CYP2C9
SCHEMBL6728842 0.85 PTGS2 (0.61) PTGS2PTGS1CYP2C9CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316485-B1 INHIBITS ACTIVITY OF CYCLOOXYGENASE-2; FOR THERAPY AND PROPHYLAXIS OF INFLAMMATION, THROMBOSIS, RHEUMATOID ARTHRITIS, ALZHEIMER'S DISEASE; AS ANALGESIC FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-13 US disclosed
EP-1017678-A1 1,5-DIPHENYLPYRAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-07-12 EP disclosed
WO-1999015505-A1 1,5-DIPHENYLPYRAZOLE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-04-01 WO disclosed