SCHEMBL7876466

SCHEMBL7876466

CC(C)NC1(C(N)=O)CC[N]CC1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
CYP2D6 P10635 1/20 0.46
KDM4E B2RXH2 1/20 0.36
KMT2A Q03164 1/20 0.36
EPHX1 P07099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12258804 0.86 ALDH1A1 (0.51) ALDH1A1CYP2D6KDM4EKMT2AEPHX1
SCHEMBL8193648 0.84 ALDH1A1 (0.50) ALDH1A1CYP2D6KDM4EKMT2A
SCHEMBL12870586 0.84 ALDH1A1 (0.50) ALDH1A1CYP2D6KDM4EKMT2A
SCHEMBL12869546 0.82 ALDH1A1 (0.49) ALDH1A1CYP2D6KDM4EKMT2A
SCHEMBL7870008 0.78 KDM4E (0.59) KDM4EKMT2A
SCHEMBL5240027 0.77 KDM4E (0.63) ALDH1A1CYP2D6KDM4EKMT2A
SCHEMBL8437435 0.76 ALDH1A1 (0.55) ALDH1A1CYP2D6KDM4EKMT2A
SCHEMBL4833027 0.72 KDM4E (0.42) ALDH1A1CYP2D6KDM4EKMT2A
SCHEMBL21916515 0.72 ALDH1A1 (0.41) ALDH1A1CYP2D6KDM4EKMT2A
SCHEMBL15461451 0.72 ALDH1A1 (0.41) ALDH1A1CYP2D6KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808303-B1 5-(4-SUBST.-PIPERIDINYL-1)-3-ARYL-PENTANOIC ACID DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONIST ASTRAZENECA AB (SE) 2001-06-20 EP disclosed
EP-0808303-A1 5-(4-SUBST.-PIPERIDINYL-1)-3-ARYL-PENTANOIC ACID DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONIST ZENECA LIMITED (GB) 1997-11-26 EP disclosed
WO-1996024582-A1 5-(4-SUBST.-PIPERIDINYL-1)-3-ARYL-PENTANOIC ACID DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONIST ZENECA LIMITED (GB) 1996-08-15 WO disclosed