SCHEMBL7878192

SCHEMBL7878192

CCOC(=O)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C(=O)N[C@H](C(=O)NC/C=C(\Cl)S(C)(=O)=O)C(C)C)c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 15/20 0.68
CASP7 P55210 10/20 0.68
CASP9 P55211 6/20 0.68
CASP10 Q92851 3/20 0.68
CASP1 P29466 7/20 0.58
CASP4 P49662 3/20 0.58
CASP8 Q14790 2/20 0.57
CASP5 P51878 1/20 0.42
CASP6 P55212 1/20 0.42
CTSB P07858 1/20 0.42
CTSK P43235 1/20 0.42
CA2 P00918 1/20 0.41
CA5A P35218 1/20 0.41
CTSL P07711 1/20 0.41
CTSS P25774 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7888193 0.93 CASP3 (0.60) CASP3CASP7CASP9CASP10CASP1
SCHEMBL7888146 0.90 CASP3 (0.55) CASP3CASP7CASP9CASP10CASP1
SCHEMBL9962260 0.89 CASP3 (0.83) CASP3CASP7CASP9CASP10CASP1
SCHEMBL7882800 0.88 CASP3 (0.66) CASP3CASP7CASP9CASP10CASP1
SCHEMBL9961964 0.87 CASP3 (0.88) CASP3CASP7CASP9CASP10CASP1
SCHEMBL9961999 0.86 CASP3 (0.88) CASP3CASP7CASP9CASP10CASP1
SCHEMBL9962320 0.86 CASP3 (0.75) CASP3CASP7CASP9CASP10CASP1
SCHEMBL7886082 0.86 CASP3 (0.59) CASP3CASP7CASP9CASP10CASP1
SCHEMBL9962316 0.84 CASP3 (0.72) CASP3CASP7CASP9CASP10CASP1
SCHEMBL7889716 0.83 CASP3 (0.65) CASP3CASP7CASP9CASP10CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010133000-A1 SELECTIVE CASPASE INHIBITORS AND USES THEREOF NEW WORLD LABORATORIES INC. (CA) 2010-11-25 WO disclosed