SCHEMBL7878503

SCHEMBL7878503

ON=C1CCOc2ccc(Cl)cc21

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.62
NPSR1 Q6W5P4 1/20 0.62
HTT P42858 2/20 0.51
PIK3CA P42336 3/20 0.43
PIK3CB P42338 3/20 0.43
PIK3CG P48736 3/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
LMNA P02545 1/20 0.40
PIK3CD O00329 1/20 0.39
MAP3K14 Q99558 1/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
NOTUM Q6P988 1/20 0.37
MAPT P10636 1/20 0.37
PKM P14618 1/20 0.37
MAOB P27338 2/20 0.36
CYP19A1 P11511 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7878501 1.00 CTSL (0.62) CTSLNPSR1HTTPIK3CAPIK3CB
SCHEMBL29991312 1.00 CTSL (0.62) CTSLNPSR1HTTPIK3CAPIK3CB
SCHEMBL11567530 0.90 CTSL (0.56) CTSLNPSR1HTTPIK3CAPIK3CB
SCHEMBL11567532 0.90 CTSL (0.56) CTSLNPSR1HTTPIK3CAPIK3CB
SCHEMBL20205932 0.83 NPSR1 (0.62) CTSLNPSR1PIK3CAPIK3CBPIK3CG
SCHEMBL13114090 0.83 NPSR1 (0.58) CTSLNPSR1PIK3CAPIK3CBPIK3CG
SCHEMBL11743822 0.80 PIK3CA (0.43) CTSLNPSR1PIK3CAPIK3CBPIK3CG
SCHEMBL17018289 0.80 MAPT (0.43) CTSLNPSR1HTTPIK3CAPIK3CB
SCHEMBL11743813 0.80 PIK3CA (0.43) CTSLNPSR1PIK3CAPIK3CBPIK3CG
SCHEMBL16997490 0.80 MAPT (0.43) CTSLNPSR1HTTPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0856514-B1 8-substituted-1,3,8-triazaspiro[4.5]decan-4-on derivatives HOFFMANN LA ROCHE (CH) 2001-06-13 EP disclosed
EP-0856514-A1 8-substituted-1,3,8-triazaspiro[4.5]decan-4-on derivatives F. HOFFMANN-LA ROCHE AG (CH) 1998-08-05 EP disclosed
US-4169097-A GASTRIC ANTISECRETORY AGENTS MORTON-NORWICH PRODUCTS, INC. (US) 1979-09-25 US disclosed