SCHEMBL7878634

SCHEMBL7878634

CNc1cccnc1Nc1cccc(CN(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.46
MEN1 O00255 5/20 0.39
KMT2A Q03164 5/20 0.39
ALDH1A1 P00352 4/20 0.39
MAPT P10636 3/20 0.39
POLB P06746 2/20 0.39
LMNA P02545 3/20 0.39
PKM P14618 2/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
GMNN O75496 1/20 0.36
TTR P02766 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
NFKB1 P19838 1/20 0.36
UGT1A1 P22309 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
PMP22 Q01453 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7880761 0.90 BRD4 (0.44) BRD4MEN1KMT2AALDH1A1MAPT
SCHEMBL7880703 0.87 BRD4 (0.44) BRD4MEN1KMT2AALDH1A1MAPT
SCHEMBL7880521 0.83 MAPT (0.48) BRD4MEN1KMT2AALDH1A1MAPT
SCHEMBL7883323 0.75 HSF1 (0.46) BRD4MAPTMAPK1GRM2
SCHEMBL7878632 0.75 LMNA (0.47) BRD4MEN1KMT2AALDH1A1MAPT
SCHEMBL7880733 0.74 FLT1 (0.41) BRD4MAPTEGFRITKNPC1
SCHEMBL7876720 0.74 BRD4 (0.45) BRD4MEN1KMT2AALDH1A1MAPT
SCHEMBL7880695 0.73 CYP3A4 (0.41) BRD4CYP1A2CYP3A4EGFRGRM2
SCHEMBL6690431 0.73 BACE1 (0.41) MEN1KMT2AMAPTNPC1RAB9A
SCHEMBL6677790 0.71 ALDH1A1 (0.47) KMT2AALDH1A1POLBCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6331553-B1 INHIBITORS OF NITRIC OXIDE SYNTHASE; TREATING CEREBROVASCULAR DISEASES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-12-18 US disclosed
EP-0949242-A1 AROMATIC AMINE DERIVATIVES HAVING NOS INHIBITORY EFFECT Chugai Seiyaku Kabushiki Kaisha (JP) 1999-10-13 EP disclosed