SCHEMBL7879263

SCHEMBL7879263

C[C@H](CCNC(=O)c1ccnnc1)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 8/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HCAR2 Q8TDS4 1/20 0.45
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
RAB9A P51151 3/20 0.43
NPC1 O15118 2/20 0.43
GRM5 P41594 1/20 0.43
TSHR P16473 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PIK3CD O00329 1/20 0.40
LMNA P02545 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15738287 0.87 SMN1; SMN2 (0.54) EPHX2CYP2C9CYP2C19HCAR2HDAC3
SCHEMBL27790062 0.79 EPHX2 (0.65) EPHX2CYP2C9CYP2C19HDAC3HDAC1
SCHEMBL10245905 0.76 NAAA (0.60) HCAR2HDAC3HDAC1SMN1; SMN2RAB9A
SCHEMBL27634018 0.75 KDM4E (0.54) EPHX2CYP2C19HDAC3HDAC1SMN1; SMN2
SCHEMBL13101050 0.75 PREP (0.45) HCAR2HDAC3HDAC1NPC1TSHR
SCHEMBL22322564 0.74 HCAR2 (0.52) HCAR2SMN1; SMN2PIK3CDLMNAMEN1
SCHEMBL31087408 0.74 RAB9A (0.70) EPHX2HDAC3HDAC1SMN1; SMN2RAB9A
SCHEMBL13113096 0.72 HCAR2 (0.48) HCAR2HDAC3HDAC1SMN1; SMN2NPC1
SCHEMBL7875218 0.71 SMN1; SMN2 (0.43) EPHX2CYP2C9CYP2C19SMN1; SMN2RAB9A
SCHEMBL21431437 0.71 CA12 (0.50) HCAR2HDAC3HDAC1LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010136474-A2 SUBSTITUTED AMINOBUTYRIC DERIVATIVES AS NEPRILYSIN INHIBITORS NOVARTIS AG (CH) 2010-12-02 WO disclosed