SCHEMBL7880720

SCHEMBL7880720

CCc1ccc(Nc2cc(C)ccn2)cc1CN

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.44
SMN1; SMN2 Q16637 6/20 0.44
NPC1 O15118 5/20 0.44
RAB9A P51151 5/20 0.44
TP53 P04637 3/20 0.44
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 1/20 0.43
KARS1 Q15046 4/20 0.43
GBA1 P04062 1/20 0.42
CYP1A2 P05177 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C19 P33261 1/20 0.42
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
LMNA P02545 1/20 0.40
NOS2 P35228 1/20 0.39
TNNI3K Q59H18 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7872384 0.84 KARS1 (0.43) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL7872421 0.84 LMNA (0.47) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL7880185 0.75 KARS1 (0.63) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL21281905 0.74 MAPK10 (0.50) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL7872531 0.74 KARS1 (0.55) SMN1; SMN2NPC1RAB9AKMT2AKARS1
SCHEMBL2912518 0.72 KDR (0.57) SMN1; SMN2NPC1RAB9AALDH1A1KMT2A
SCHEMBL18772775 0.72 TNNI3K (0.59) SMN1; SMN2NPC1RAB9ATP53KMT2A
SCHEMBL7878698 0.71 KARS1 (0.49) NPC1ALDH1A1KMT2AKARS1KDM4E
SCHEMBL7880192 0.70 KARS1 (0.48) NPC1KMT2AKARS1NOS2
SCHEMBL27524202 0.70 KARS1 (0.48) NPC1ALDH1A1KMT2AKARS1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1244542-C Aromatic amine derivatives having NOS inhibitory effect CHUGAI PHARMACEUTICAL CO LTD (JP) 2006-03-08 CN claimed
US-6331553-B1 INHIBITORS OF NITRIC OXIDE SYNTHASE; TREATING CEREBROVASCULAR DISEASES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-12-18 US claimed
CN-1240419-A Aromatic amine derivatives having NOS inhibitory effect CHUGAI PHARMACEUTICAL CO LTD (JP) 2000-01-05 CN claimed
EP-0949242-A1 AROMATIC AMINE DERIVATIVES HAVING NOS INHIBITORY EFFECT Chugai Seiyaku Kabushiki Kaisha (JP) 1999-10-13 EP claimed
CN-1244542-C Aromatic amine derivatives having NOS inhibitory effect CHUGAI PHARMACEUTICAL CO LTD (JP) 2006-03-08 CN disclosed
US-6331553-B1 INHIBITORS OF NITRIC OXIDE SYNTHASE; TREATING CEREBROVASCULAR DISEASES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-12-18 US disclosed
CN-1240419-A Aromatic amine derivatives having NOS inhibitory effect CHUGAI PHARMACEUTICAL CO LTD (JP) 2000-01-05 CN disclosed
EP-0949242-A1 AROMATIC AMINE DERIVATIVES HAVING NOS INHIBITORY EFFECT Chugai Seiyaku Kabushiki Kaisha (JP) 1999-10-13 EP disclosed