SCHEMBL7880947

SCHEMBL7880947

O=C(O)CCc1c[nH]c2c1CCC=C2

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPR17 Q13304 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPSR1 Q6W5P4 1/20 0.35
PARP1 P09874 1/20 0.33
ADORA3 P0DMS8 1/20 0.30
PDGFRB P09619 1/20 0.30
FGFR1 P11362 1/20 0.30
KDR P35968 1/20 0.30
ZAP70 P43403 1/20 0.30
KEAP1 Q14145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12536197 0.79 KDM4E (0.41) HPGD
SCHEMBL14300543 0.78 HTR2A (0.35) PARP1
SCHEMBL7051131 0.77
SCHEMBL6299779 0.70 NPSR1 (0.42) GPR17HPGDCYP2C19NPSR1PARP1
SCHEMBL6691776 0.69 NPSR1 (0.41) GPR17HPGDCYP2C19NPSR1PARP1
SCHEMBL13542070 0.64
SCHEMBL28737712 0.64 NPSR1 (0.54) GPR17HPGDCYP2C19NPSR1PARP1
SCHEMBL18738896 0.64 GPR17 (0.38) GPR17HPGDCYP2C19NPSR1PARP1
SCHEMBL1171886 0.61 NPSR1 (0.52) GPR17HPGDCYP2C19NPSR1PARP1
SCHEMBL3797505 0.61 GPR17 (0.40) GPR17HPGDCYP2C19NPSR1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010136474-A2 SUBSTITUTED AMINOBUTYRIC DERIVATIVES AS NEPRILYSIN INHIBITORS NOVARTIS AG (CH) 2010-12-02 WO disclosed
WO-2008005368-A2 PIPERAZINES AS P2X7 ANTAGONISTS ABBOTT LABORATORIES (US) 2008-01-10 WO disclosed