SCHEMBL7883448

SCHEMBL7883448

Bc1c(C2CCC(C(=O)O)CC2)nc2c(-c3ccc(-c4ccc(F)c(F)c4)nc3)cnn2c1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 11/20 0.42
KCNH2 Q12809 3/20 0.38
MTOR P42345 3/20 0.37
RPTOR Q8N122 3/20 0.37
MLST8 Q9BVC4 3/20 0.37
SOAT1 P35610 1/20 0.36
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PARP1 P09874 1/20 0.33
GRIN2B Q13224 1/20 0.33
CHEK1 O14757 2/20 0.33
CCNA2 P20248 2/20 0.33
CDK2 P24941 2/20 0.33
CCNA1 P78396 2/20 0.33
IGF1R P08069 1/20 0.33
ADORA2A P29274 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10236821 0.90 CHEK1 (0.44) DGAT1KCNH2MTORRPTORMLST8
SCHEMBL7886219 0.88 DGAT1 (0.39) DGAT1KCNH2MTORRPTORMLST8
SCHEMBL7874478 0.87 MTOR (0.40) DGAT1KCNH2MTORRPTORMLST8
SCHEMBL10234279 0.83 CHEK1 (0.44) DGAT1KCNH2MTORRPTORMLST8
SCHEMBL10234251 0.81 CHEK1 (0.46) DGAT1MTORRPTORMLST8CHEK1
SCHEMBL7885498 0.81 CHEK1 (0.46) DGAT1MTORRPTORMLST8CHEK1
SCHEMBL7875038 0.80 CHEK1 (0.46) DGAT1MTORRPTORMLST8KDM4E
SCHEMBL7882451 0.79 MTOR (0.43) MTORRPTORMLST8KDM4ENPC1
SCHEMBL7874817 0.79 MTOR (0.44) MTORRPTORMLST8KDM4ENPC1
SCHEMBL7882513 0.79 KMT2A (0.40) DGAT1MTORRPTORMLST8KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118207-A1 PYRAZOLO [1, 5-A] PYRIMIDINE DERIVATIVES AS MTOR INHIBITORS SCHERING CORPORATION (US) 2010-10-14 WO disclosed