SCHEMBL7885162

SCHEMBL7885162

Brc1cccc(NOc2ccccc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.50
ALDH1A1 P00352 4/20 0.49
MEN1 O00255 2/20 0.49
KDM4E B2RXH2 2/20 0.49
LMNA P02545 1/20 0.46
HPGD P15428 1/20 0.46
ALOX12 P18054 1/20 0.46
MAOB P27338 3/20 0.44
PGR P06401 1/20 0.42
ABCB1 P08183 1/20 0.41
ABCC1 P33527 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41
MAOA P21397 1/20 0.41
FAAH O00519 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
HTT P42858 1/20 0.40
IDO1 P14902 1/20 0.40
RAPGEF4 Q8WZA2 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
P2RX1 P51575 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7885157 0.89 KMT2A (0.54) KMT2AALDH1A1MEN1KDM4ELMNA
SCHEMBL251644 0.79 ALDH1A1 (0.43) KMT2AALDH1A1MEN1KDM4ELMNA
SCHEMBL1283693 0.78 ALDH1A1 (0.44) KMT2AALDH1A1MEN1LMNAHPGD
SCHEMBL1964058 0.77 ALDH1A1 (0.42) KMT2AALDH1A1MEN1KDM4ELMNA
SCHEMBL633344 0.77 HTT (0.54) KMT2AALDH1A1MEN1LMNAHPGD
SCHEMBL15839989 0.77 MEN1 (0.57) KMT2AALDH1A1MEN1KDM4ELMNA
SCHEMBL14071502 0.75 KMT2A (0.50) KMT2AALDH1A1MEN1KDM4ELMNA
SCHEMBL10961976 0.74 CYP2A6 (0.50) KMT2AALDH1A1MEN1KDM4ELMNA
SCHEMBL19411968 0.74 ALDH1A1 (0.43) KMT2AALDH1A1MEN1KDM4ELMNA
SCHEMBL1187729 0.74 GAA (0.50) KMT2AALDH1A1MEN1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147093-A1 SUBSTITUTED BICYCLIC DERIVATIVES USEFUL AS ANTICANCER AGENTS Pfizer Products Inc. (US) 2001-10-24 EP disclosed
WO-2000044728-A1 SUBSTITUTED BICYCLIC DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PRODUCTS INC. (US) 2000-08-03 WO disclosed