SCHEMBL7889207

SCHEMBL7889207

COc1ccc2c(c1)CCN(S(=O)(=O)c1ccc(C)cc1)[C@@H](C)[C@@H]2O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
CA1 P00915 4/20 0.55
CA2 P00918 4/20 0.55
CA9 Q16790 4/20 0.55
CA14 Q9ULX7 4/20 0.55
TAS2R14 Q9NYV8 2/20 0.54
MMP1 P03956 5/20 0.52
MMP2 P08253 5/20 0.52
MMP9 P14780 5/20 0.52
MMP12 P39900 5/20 0.52
MMP14 P50281 5/20 0.52
MMP15 P51511 5/20 0.52
MMP16 P51512 5/20 0.52
MMP26 Q9NRE1 5/20 0.52
MMP7 P09237 4/20 0.49
CA7 P43166 1/20 0.49
LMNA P02545 2/20 0.47
MAPT P10636 1/20 0.47
ESR1 P03372 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3394741 0.84 MMP1 (0.70) MEN1KMT2ATAS2R14MMP1MMP2
SCHEMBL3397104 0.84 MMP1 (0.70) MEN1KMT2ATAS2R14MMP1MMP2
SCHEMBL3392159 0.84 MMP1 (0.70) MEN1KMT2ATAS2R14MMP1MMP2
SCHEMBL3393324 0.84 MMP1 (0.70) MEN1KMT2ATAS2R14MMP1MMP2
SCHEMBL3397077 0.79 RYR2 (0.51) MEN1KMT2ACA1CA2CA9
SCHEMBL29052386 0.78 MEN1 (0.57) MEN1KMT2ACA1CA2CA9
SCHEMBL3393154 0.76 MEN1 (0.60) MEN1KMT2ACA1CA2CA9
SCHEMBL3393158 0.76 MEN1 (0.60) MEN1KMT2ACA1CA2CA9
SCHEMBL29051730 0.76 CA1 (0.48) MEN1KMT2ACA1CA2CA9
SCHEMBL1016818 0.72 PKM (0.62) MEN1KMT2ALMNARYR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246331-A1 NR2B-selective NMDA-receptor antagonists Westfälische Wilhelms-Universität Münster (DE) 2010-11-03 EP disclosed
WO-2010122134-A1 NR2B-SELECTIVE NMDA-RECEPTOR ANTAGONISTS Westfälische Wilhelms Universität Münster (DE) 2010-10-28 WO disclosed