SCHEMBL7889384

SCHEMBL7889384

Cc1cc(C(=O)NCc2cccc([N+](=O)[O-])c2)c(NC(=O)c2ccc(C(=O)O)cc2)s1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
MAPT P10636 3/20 0.56
SMN1; SMN2 Q16637 1/20 0.52
ACKR3 P25106 1/20 0.51
SENP5 Q96HI0 3/20 0.48
SENP2 Q9HC62 3/20 0.48
SENP1 Q9P0U3 3/20 0.48
FFAR1 O14842 1/20 0.47
LMNA P02545 2/20 0.46
AKR1B1 P15121 1/20 0.46
OPRM1 P35372 1/20 0.46
OPRK1 P41145 1/20 0.46
PPARG P37231 1/20 0.44
HPGD P15428 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
RECQL P46063 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8210314 0.91 ALDH1A1 (0.48) ALDH1A1MAPTSMN1; SMN2ACKR3SENP5
SCHEMBL7889261 0.89 ALDH1A1 (0.55) ALDH1A1MAPTSMN1; SMN2ACKR3SENP5
SCHEMBL8209703 0.89 ALDH1A1 (0.56) ALDH1A1MAPTSMN1; SMN2ACKR3SENP5
SCHEMBL7888341 0.86 NR1H4 (0.50) ALDH1A1MAPTSMN1; SMN2LMNAHPGD
SCHEMBL7430376 0.81 ACKR3 (0.48) ALDH1A1MAPTSMN1; SMN2ACKR3SENP5
SCHEMBL8212457 0.81 AKR1B1 (0.49) ALDH1A1MAPTSMN1; SMN2ACKR3SENP5
Bicarbonate SCHEMBL7430381 0.81 POLB (0.48) ALDH1A1MAPTSMN1; SMN2ACKR3SENP5
SCHEMBL8207378 0.80 ALDH1A1 (0.48) ALDH1A1MAPTSMN1; SMN2ACKR3SENP5
SCHEMBL8211512 0.79 ACKR3 (0.55) ALDH1A1MAPTACKR3LMNAAKR1B1
SCHEMBL7892988 0.79 NR1H4 (0.58) ALDH1A1MAPTSMN1; SMN2HPGDRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934301-B1 AMINOTHIOPHENE CARBOXYLIC ACID AMIDES AND THE USE THEREOF AS PHOSPHODIESTERASE INHIBITORS MERCK PATENT GMBH (DE) 2001-06-20 EP disclosed
US-6143777-A ENZYME INHIBITORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-07 US disclosed