SCHEMBL7891103

SCHEMBL7891103

COC(=O)[C@H](C)N(CCc1cccc(OC)c1)S(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BMP1 P13497 3/20 0.53
L3MBTL1 Q9Y468 1/20 0.49
PTGER1 P34995 1/20 0.48
TAS2R14 Q9NYV8 3/20 0.47
TP53 P04637 2/20 0.46
PKM P14618 1/20 0.45
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA9 Q16790 2/20 0.44
AKR1C3 P42330 1/20 0.44
CA7 P43166 1/20 0.44
CA14 Q9ULX7 1/20 0.44
CA12 O43570 1/20 0.44
CA4 P22748 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13069327 0.91 KEAP1 (0.54) BMP1L3MBTL1PTGER1TAS2R14TP53
SCHEMBL7889204 0.89 CA12 (0.47) BMP1TP53CA1CA2CA9
SCHEMBL7879881 0.89 CA12 (0.47) BMP1TP53CA1CA2CA9
SCHEMBL3811847 0.82 BMP1 (0.50) BMP1L3MBTL1PTGER1TAS2R14TP53
SCHEMBL3398501 0.82 BMP1 (0.50) BMP1L3MBTL1PTGER1TAS2R14TP53
SCHEMBL29051740 0.81 PTGER1 (0.48) BMP1L3MBTL1PTGER1TAS2R14PKM
SCHEMBL29051743 0.81 PTGER1 (0.48) BMP1L3MBTL1PTGER1TAS2R14PKM
SCHEMBL3393112 0.80 CA12 (0.49) CA1CA2CA9CA12CA4
SCHEMBL3393113 0.80 CA12 (0.49) CA1CA2CA9CA12CA4
SCHEMBL7888158 0.80 CA12 (0.49) CA1CA2CA9CA12CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2246331-A1 NR2B-selective NMDA-receptor antagonists Westfälische Wilhelms-Universität Münster (DE) 2010-11-03 EP disclosed
WO-2010122134-A1 NR2B-SELECTIVE NMDA-RECEPTOR ANTAGONISTS Westfälische Wilhelms Universität Münster (DE) 2010-10-28 WO disclosed