SCHEMBL7894512

SCHEMBL7894512

CCOC(=O)C(CC(=O)O)=C(c1ccc(S(C)(=O)=O)cc1)c1cccc(Br)c1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.51
PTGS2 P35354 8/20 0.48
AKR1C3 P42330 1/20 0.46
AKR1C2 P52895 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7894510 1.00 CYP19A1 (0.51) CYP19A1PTGS2AKR1C3AKR1C2
SCHEMBL7898781 0.91 NHERF1 (0.47) CYP19A1PTGS2AKR1C3
SCHEMBL7898784 0.91 NHERF1 (0.47) CYP19A1PTGS2AKR1C3
SCHEMBL8155346 0.91 PTGS2 (0.53) CYP19A1PTGS2
SCHEMBL8155347 0.91 PTGS2 (0.53) CYP19A1PTGS2
SCHEMBL7895226 0.90 PTGS2 (0.45) CYP19A1PTGS2
SCHEMBL7895227 0.90 PTGS2 (0.45) CYP19A1PTGS2
SCHEMBL7894395 0.88 AKR1C3 (0.45) PTGS2AKR1C3
SCHEMBL7894390 0.88 AKR1C3 (0.45) PTGS2AKR1C3
SCHEMBL7898845 0.88 AKR1C3 (0.47) CYP19A1PTGS2AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6180651-B1 ANTIINFLAMMATORY AGENTS; ANALGESICS BRISTOL-MYERS SQUIBB 2001-01-30 US disclosed
WO-2000014082-A1 DIARYLMETHYLIDENE FURAN DERIVATIVES AS DRUGS WITH ANTI-INFLAMMATORY, ANALGESIC AND CHEMOPREVENTIVE PROPERTIES LABORATORIES UPSA (FR) 2000-03-16 WO disclosed
US-5807873-A Diarylmethylidenefuran derivatives and their uses in therapeutics LABORATORIES UPSA (FR) 1998-09-15 US disclosed