SCHEMBL7894993

SCHEMBL7894993

CC(Nc1c(NCc2ccc(C#N)c(Cl)c2)c(=O)c1=O)C(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 1/20 0.47
ABCC8 Q09428 1/20 0.47
KCNJ11 Q14654 1/20 0.47
KCNJ8 Q15842 1/20 0.47
PLK1 P53350 5/20 0.40
CHEK1 O14757 3/20 0.40
ROCK2 O75116 3/20 0.40
CHEK2 O96017 3/20 0.40
GSK3A P49840 3/20 0.40
GSK3B P49841 3/20 0.40
ROCK1 Q13464 3/20 0.40
PKN2 Q16513 3/20 0.40
CDC42BPA Q5VT25 3/20 0.40
CSNK1G3 Q9Y6M4 3/20 0.40
PIM1 P11309 2/20 0.40
PRKX P51817 2/20 0.40
CSNK1G2 P78368 2/20 0.40
PLK3 Q9H4B4 2/20 0.40
CLK4 Q9HAZ1 2/20 0.40
MKNK2 Q9HBH9 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7895070 0.86 ABCC9 (0.55) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL7895708 0.83 PLK1 (0.42) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL7895472 0.83 CHEK2 (0.43) CHEK1ROCK2CHEK2GSK3AGSK3B
SCHEMBL8370799 0.81 PLK1 (0.54) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL8370803 0.81 PLK1 (0.54) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL7886866 0.80 ABCC9 (0.58) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL7894022 0.80 ABCC9 (0.58) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL7886860 0.80 ABCC9 (0.58) ABCC9ABCC8KCNJ11KCNJ8PLK1
SCHEMBL7894223 0.80 CHEK2 (0.41) CHEK1ROCK2CHEK2GSK3AGSK3B
SCHEMBL7895113 0.77 ABCC9 (0.60) ABCC9ABCC8KCNJ11KCNJ8PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1151990-A1 Substituted N-arylmethylamino derivatives of cyclobutene-3, 4-diones AMERICAN HOME PRODUCTS CORPORATION (US) 2001-11-07 EP claimed
US-5780505-A ADMINISTERING AS SMOOTH MUSCLE RELAXANT AMERICAN HOME PRODUCTS CORPORATION (US) 1998-07-14 US claimed
EP-1151990-A1 Substituted N-arylmethylamino derivatives of cyclobutene-3, 4-diones AMERICAN HOME PRODUCTS CORPORATION (US) 2001-11-07 EP disclosed