SCHEMBL7895228

SCHEMBL7895228

c1cnc(N2CCC3(CC2)c2ccccc2CCn2ccnc23)nc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.47
OPRK1 P41145 1/20 0.47
HRH1 P35367 2/20 0.39
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
CYP3A4 P08684 4/20 0.37
CYP2D6 P10635 2/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
ALDH1A1 P00352 3/20 0.36
SIGMAR1 Q99720 3/20 0.35
CYP2C9 P11712 2/20 0.34
MAPK1 P28482 2/20 0.34
DRD3 P35462 2/20 0.34
MEN1 O00255 2/20 0.34
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP2C19 P33261 2/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6031086 0.82 HRH1 (0.54) HRH1CYP3A4CYP2D6TSHRSMN1; SMN2
Hydrochloric Acid SCHEMBL6030477 0.81 HRH1 (0.55) HRH1CYP3A4CYP2D6TSHRSMN1; SMN2
SCHEMBL6030048 0.81 SIGMAR1 (0.43) HRH1SIGMAR1
SCHEMBL6030987 0.80 SIGMAR1 (0.53) OPRD1OPRK1CYP3A4CYP2D6TSHR
SCHEMBL6031884 0.79 SIGMAR1 (0.37) HRH1CYP3A4CYP2D6TSHRALDH1A1
SCHEMBL6031686 0.78 SIGMAR1 (0.55) SIGMAR1
Hydrochloric Acid SCHEMBL6100154 0.77 SIGMAR1 (0.38) HRH1SIGMAR1
Iodide SCHEMBL6031820 0.75 SIGMAR1 (0.56) OPRD1OPRK1HRH1SIGMAR1
Isopropyl Alcohol SCHEMBL6101083 0.75 SIGMAR1 (0.39) HRH1SIGMAR1
SCHEMBL6030965 0.75 OPRD1 (0.55) OPRD1OPRK1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144411-A1 ANTIHISTAMINIC SPIRO COMPOUNDS Janssen Pharmaceutica N.V. (BE) 2001-10-17 EP disclosed
WO-2000037470-A1 ANTIHISTAMINIC SPIRO COMPOUNDS JANSSEN PHARMACEUTICA N.V. (BE) 2000-06-29 WO disclosed