SCHEMBL7895618

SCHEMBL7895618

CC(C)C(C)Nc1c(NCc2ccc(C#N)cc2)c(=O)c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 2/20 0.47
ABCC9 O60706 1/20 0.43
ABCC8 Q09428 1/20 0.43
KCNJ11 Q14654 1/20 0.43
KCNJ8 Q15842 1/20 0.43
CYP19A1 P11511 1/20 0.40
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
CYP2A6 P11509 1/20 0.39
CHEK1 O14757 2/20 0.38
CHEK2 O96017 2/20 0.38
PRKACA P17612 2/20 0.38
RPS6KB1 P23443 2/20 0.38
GSK3A P49840 2/20 0.38
GSK3B P49841 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7894087 0.88 LOXL2 (0.50) LOXL2ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL7886860 0.86 ABCC9 (0.58) LOXL2ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL7894022 0.86 ABCC9 (0.58) LOXL2ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL7886866 0.86 ABCC9 (0.58) LOXL2ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL7886885 0.84 LOXL2 (0.46) LOXL2ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL7886886 0.84 LOXL2 (0.46) LOXL2ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL7887143 0.83 LOXL2 (0.47) LOXL2ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL7887274 0.82 LOXL2 (0.50) LOXL2ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL7894067 0.80 LOXL2 (0.59) LOXL2CYP19A1KDM4EALDH1A1CYP1A2
SCHEMBL8373578 0.79 ABCC9 (0.47) ABCC9ABCC8KCNJ11KCNJ8CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1151990-A1 Substituted N-arylmethylamino derivatives of cyclobutene-3, 4-diones AMERICAN HOME PRODUCTS CORPORATION (US) 2001-11-07 EP claimed
US-5846999-A Substituted N-arylmethylamino derivatives of cyclobutene-3,4-diones AMERICAN HOME PRODUCTS CORPORATION (US) 1998-12-08 US claimed
EP-1151990-A1 Substituted N-arylmethylamino derivatives of cyclobutene-3, 4-diones AMERICAN HOME PRODUCTS CORPORATION (US) 2001-11-07 EP disclosed
US-5846999-A Substituted N-arylmethylamino derivatives of cyclobutene-3,4-diones AMERICAN HOME PRODUCTS CORPORATION (US) 1998-12-08 US disclosed