SCHEMBL789969

SCHEMBL789969

Cc1ccc(Nc2nc(CN3CCC(C)CC3)c(C)s2)c(C)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.45
ALDH1A1 P00352 5/20 0.45
NPC1 O15118 4/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
MAPT P10636 3/20 0.45
POLB P06746 2/20 0.45
LMNA P02545 4/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
MAPK1 P28482 2/20 0.42
ALOX15 P16050 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KDM4E B2RXH2 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ACHE P22303 2/20 0.38
OPRM1 P35372 1/20 0.38
TSHR P16473 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL789561 0.81 TRPC3 (0.42) RAB9AALDH1A1SMN1; SMN2MAPTLMNA
SCHEMBL12503735 0.76 TRPC3 (0.48) RAB9AALDH1A1NPC1SMN1; SMN2MAPT
SCHEMBL806645 0.66 TRPC3 (0.58) ALDH1A1SMN1; SMN2MAPTTP53
SCHEMBL17828172 0.63 KCNH2 (0.47) RAB9AALDH1A1NPC1SMN1; SMN2L3MBTL1
SCHEMBL8048110 0.62 SMN1; SMN2 (0.51) RAB9AALDH1A1NPC1SMN1; SMN2MAPT
SCHEMBL8275450 0.61 HRH3 (0.76) ALDH1A1POLBLMNAL3MBTL1ACHE
SCHEMBL12749634 0.61 NPC1 (1.00) RAB9AALDH1A1NPC1SMN1; SMN2MAPT
SCHEMBL15214324 0.61 TSHR (0.59) RAB9AALDH1A1NPC1MAPTMAPK1
SCHEMBL27954331 0.60 NPC1 (0.41) RAB9AALDH1A1NPC1SMN1; SMN2MAPT
SCHEMBL156415 0.60 ACHE (0.67) ALDH1A1MAPTKDM4EACHEMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037351-A1 COMPOUNDS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed