SCHEMBL7900098

SCHEMBL7900098

O=C(O)CC1NC(=O)OC1c1ccc(Br)cc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
GAA P10253 1/20 0.35
HDAC4 P56524 1/20 0.35
MDM2 Q00987 3/20 0.35
ALDH1A1 P00352 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
GRM5 P41594 1/20 0.33
APEX1 P27695 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7900105 0.83 EGFR (0.39) KMT2AMEN1GAAMDM2ALDH1A1
SCHEMBL7899177 0.78 CYP2C9 (0.43) CYP2C9CYP2C19KMT2AMEN1GAA
SCHEMBL15676054 0.73 GRM5 (0.45) CYP2C9CYP2C19ALDH1A1GRM5KDM4E
SCHEMBL19795867 0.73 GRM5 (0.45) CYP2C9CYP2C19ALDH1A1GRM5KDM4E
SCHEMBL5136321 0.72 LMNA (0.40) CYP2C9CYP2C19KMT2AMEN1MDM2
SCHEMBL14437759 0.72 LMNA (0.40) CYP2C9CYP2C19KMT2AMEN1MDM2
SCHEMBL30695642 0.71 MDM2 (0.43) CYP2C9CYP2C19KMT2AMEN1GAA
SCHEMBL15699098 0.68 GRM5 (0.44) KMT2AMEN1GRM5
SCHEMBL15676299 0.68 GRM5 (0.44) KMT2AMEN1GRM5
SCHEMBL19061962 0.68 GRM5 (0.44) KMT2AMEN1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed