SCHEMBL7900441

SCHEMBL7900441

COc1cc(-c2cnc3[nH]c(=O)n(-c4ccc5c(c4)CCN5)c3n2)ccc1OCCN1CCOCC1

nearest known ligand 0.66

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MAP3K11 Q16584 18/20 0.66
ADORA2A P29274 2/20 0.49
LRRK2 Q5S007 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7897792 0.93 MAP3K11 (0.74) MAP3K11LRRK2
SCHEMBL723838 0.85 MAP3K11 (0.85) MAP3K11LRRK2
SCHEMBL7910405 0.83 MAP3K11 (0.62) MAP3K11LRRK2
SCHEMBL7907784 0.81 MAP3K11 (0.74) MAP3K11LRRK2
SCHEMBL7913447 0.80 MAP4K1 (0.56) MAP3K11ADORA2ALRRK2
SCHEMBL721892 0.80 MAP3K11 (1.00) MAP3K11ADORA2A
SCHEMBL721043 0.78 MAP3K11 (1.00) MAP3K11LRRK2
SCHEMBL722057 0.78 MAP3K11 (1.00) MAP3K11ADORA2A
SCHEMBL7906450 0.76 MAP3K11 (0.68) MAP3K11
SCHEMBL7910327 0.76 MAP3K11 (0.64) MAP3K11LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149950-A2 BICYCLIC HETEROARYL KINASE INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2011-12-01 WO disclosed
WO-2010068483-A2 MLK INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2010-06-17 WO disclosed