SCHEMBL7913447

SCHEMBL7913447

COc1cc(-c2cnc3[nH]cc(-c4ccc5c(c4)CCN5)c3n2)ccc1OCCN1CCOCC1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 8/20 0.56
KIT P10721 1/20 0.54
MAP3K11 Q16584 3/20 0.52
MAPK1 P28482 1/20 0.47
ADORA2A P29274 2/20 0.45
IL2 P60568 1/20 0.44
JAK2 O60674 1/20 0.44
JAK1 P23458 1/20 0.44
JAK3 P52333 1/20 0.44
PRKAB2 O43741 1/20 0.42
PRKAG1 P54619 1/20 0.42
PRKAA2 P54646 1/20 0.42
PRKAA1 Q13131 1/20 0.42
PRKAG3 Q9UGI9 1/20 0.42
PRKAG2 Q9UGJ0 1/20 0.42
PRKAB1 Q9Y478 1/20 0.42
RET P07949 1/20 0.41
LRRK2 Q5S007 1/20 0.41
CHEK1 O14757 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL722011 0.84 KIT (0.56) MAP4K1KITMAP3K11MAPK1ADORA2A
SCHEMBL7900441 0.80 MAP3K11 (0.66) MAP3K11ADORA2ALRRK2
SCHEMBL7908343 0.80 MAP4K1 (0.54) MAP4K1KITMAP3K11MAPK1
SCHEMBL7905131 0.80 MAP4K1 (0.54) MAP4K1KITMAP3K11MAPK1JAK2
SCHEMBL7905848 0.79 KIT (0.60) MAP4K1KITIL2
SCHEMBL7897792 0.73 MAP3K11 (0.74) MAP3K11LRRK2
SCHEMBL7094017 0.72 SYK (0.52) MAPK1LRRK2CHEK1
SCHEMBL2801860 0.71 JAK2 (0.59) KITMAP3K11ADORA2AJAK2JAK1
SCHEMBL12763549 0.71 KIT (0.75) MAP4K1KITMAP3K11IL2
SCHEMBL15653841 0.70 MAPK1 (0.48) MAP4K1KITMAP3K11MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010068483-A2 MLK INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2010-06-17 WO disclosed