SCHEMBL7900624

SCHEMBL7900624

C=C1C=C(C(=O)N2CCNCC2)C=CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.42
RXFP1 Q9HBX9 1/20 0.39
HPGD P15428 1/20 0.37
HSP90AA1 P07900 1/20 0.37
SETD7 Q8WTS6 1/20 0.36
SCN5A Q14524 1/20 0.36
SCN2A Q99250 1/20 0.36
SCN10A Q9Y5Y9 1/20 0.36
HRH4 Q9H3N8 3/20 0.35
HRH3 Q9Y5N1 1/20 0.35
KMT2A Q03164 1/20 0.35
TP53 P04637 1/20 0.35
MDM2 Q00987 1/20 0.35
CA2 P00918 2/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA9 Q16790 1/20 0.34
CHKA P35790 1/20 0.33
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7890961 0.78 SIGMAR1 (0.40) SIGMAR1RXFP1HPGDHSP90AA1SETD7
SCHEMBL7899238 0.72
SCHEMBL10956840 0.70
SCHEMBL7900621 0.69 SIGMAR1 (0.42) SIGMAR1RXFP1HPGDHSP90AA1SETD7
SCHEMBL6634977 0.65 SIGMAR1 (0.45) SIGMAR1RXFP1HPGDHSP90AA1SETD7
SCHEMBL8358137 0.64 SIGMAR1 (0.81) SIGMAR1RXFP1HPGDMKNK1MKNK2
SCHEMBL13295236 0.64 SIGMAR1 (0.47) SIGMAR1RXFP1HPGDHSP90AA1HRH4
SCHEMBL9396214 0.62 CA2 (0.59) SIGMAR1RXFP1HPGDHSP90AA1HRH4
SCHEMBL8253848 0.61 RXFP1 (0.77) SIGMAR1RXFP1HSP90AA1HRH4HRH3
SCHEMBL304221 0.61 SIGMAR1 (0.68) SIGMAR1RXFP1HPGDMKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191273-B1 3,6,10,14-SUBSTITUTED-3,6,10,16-TETRAAZABICYCLO(10.3.1)-HEXADE CA-1(16),12,14-TRIENE COMPOUNDS OF GIVEN FORMULA; ANTIBACTERIAL AND OTHER UTILITIES, SUCH AS TO SCREEN FOR PESTICIDES OR DRUGS ISIS PHARMACEUTICALS, INC. 2001-02-20 US disclosed
WO-1999011612-A2 SUBSTITUTED CYCLIC COMPOUNDS AND MIXTURES COMPRISING SAME ISIS PHARMACEUTICALS, INC. (US) 1999-03-11 WO disclosed