SCHEMBL7901138

SCHEMBL7901138

COc1cc(-c2c[nH]nn2)ccc1-c1ccnc(C)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 6/20 0.45
PSEN2 P49810 6/20 0.45
APH1B Q8WW43 6/20 0.45
NCSTN Q92542 6/20 0.45
APH1A Q96BI3 6/20 0.45
PSENEN Q9NZ42 6/20 0.45
DYRK1A Q13627 5/20 0.44
PIM1 P11309 1/20 0.44
DYRK2 Q92630 1/20 0.44
DYRK1B Q9Y463 1/20 0.44
S1PR1 P21453 1/20 0.42
S1PR3 Q99500 1/20 0.42
NFATC1 O95644 1/20 0.40
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40
KIT P10721 4/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
PIK3CA P42336 1/20 0.38
WNT3A P56704 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5479059 0.78 GUSB (0.42) CYP3A4CYP2D6KMT2A
SCHEMBL6915415 0.76 DYRK1A (0.49) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL12516813 0.76 DYRK1A (0.51) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL27971322 0.76 ALDH1A1 (0.56) DYRK1AKITKMT2A
SCHEMBL7896922 0.74 DYRK1A (0.49) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL29637091 0.74 DYRK1A (0.49) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1492639 0.74 DYRK1A (0.49) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL11919644 0.71 WNT3A (0.54) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2350999 0.71 DYRK1A (0.66) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2489888 0.70 ALDH1A1 (0.50) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010071741-A1 TRIAZOLE DERIVATIVES FOR TREATMENT OF ALZHEIMER'S DISEASE MERCK SHARP & DOHME CORP. (US) 2010-06-24 WO disclosed