SCHEMBL7901592

SCHEMBL7901592

COc1ccc2c(c1OC)C[C@H]1CCCN(C(=O)O)[C@@H]1C2

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.41
DRD2 P14416 5/20 0.40
DRD1 P21728 3/20 0.40
HTR1A P08908 6/20 0.40
PARP1 P09874 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7907814 1.00 HSD11B1 (0.41) HSD11B1DRD2DRD1HTR1APARP1
SCHEMBL7901664 0.90 DRD2 (0.39) HSD11B1DRD2DRD1HTR1APARP1
SCHEMBL15382598 0.87 HSD11B1 (0.39) HSD11B1DRD2DRD1HTR1APARP1
SCHEMBL50764 0.87 HSD11B1 (0.39) HSD11B1DRD2DRD1HTR1APARP1
SCHEMBL50762 0.87 HSD11B1 (0.39) HSD11B1DRD2DRD1HTR1APARP1
SCHEMBL50763 0.87 HSD11B1 (0.39) HSD11B1DRD2DRD1HTR1APARP1
SCHEMBL51067 0.87 HSD11B1 (0.39) HSD11B1DRD2DRD1HTR1APARP1
SCHEMBL21255627 0.87 HSD11B1 (0.39) HSD11B1DRD2DRD1HTR1APARP1
SCHEMBL3322834 0.82 DRD2 (0.40) DRD2DRD1HTR1A
SCHEMBL51300 0.82 DRD2 (0.56) DRD2DRD1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097091-A1 METHODS OF ADMINISTERING (4AR, 1OAR)-I-N-PROPYL-I, 2,3,4A7 S1IO7 IOA-OCTAHYDROBENZO [G] QUINOLINE-6,7-DIOL AND RELATED COMPOUNDS ACROSS THE ORAL MUCOSA, THE NASAL MUCOSA OR THE SKIN AND PHARMACEUTICAL COMPOSITIONS THEREOF H. LUNDBECK A/S (DK) 2010-09-02 WO disclosed
WO-2010097092-A1 TREATMENT OF DYSKINESIA RELATED DISORDERS H. LUNDBECK A/S (DK) 2010-09-02 WO disclosed