SCHEMBL7901625

SCHEMBL7901625

CON(C)C(=O)Nc1ccc(OCCc2ccc(C)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.51
MEN1 O00255 2/20 0.51
RAB9A P51151 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
PKM P14618 1/20 0.51
MAPT P10636 2/20 0.50
HTT P42858 2/20 0.50
HPGD P15428 1/20 0.50
KCNH2 Q12809 1/20 0.47
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
NPC1 O15118 1/20 0.46
TP53 P04637 1/20 0.46
FFAR1 O14842 2/20 0.46
PPARA Q07869 3/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
KDM4E B2RXH2 1/20 0.45
GAA P10253 1/20 0.45
PPARD Q03181 1/20 0.45
LTB4R Q15722 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9799004 1.00 KMT2A (0.51) KMT2AMEN1RAB9ATDP1PKM
SCHEMBL11657341 0.91 MEN1 (0.52) KMT2AMEN1RAB9ATDP1PKM
SCHEMBL11332580 0.89 PKM (0.68) KMT2AMEN1RAB9ATDP1PKM
SCHEMBL11270005 0.89 NPY5R (0.56) KMT2AMEN1RAB9ATDP1PKM
SCHEMBL11304645 0.88 MAPT (0.50) KMT2AMEN1RAB9AMAPTHTT
SCHEMBL11221817 0.88 MEN1 (0.60) KMT2AMEN1RAB9ATDP1PKM
SCHEMBL11572411 0.87 MAPT (0.49) KMT2AMEN1RAB9AMAPTHTT
SCHEMBL11657307 0.87 RAB9A (0.51) KMT2AMEN1RAB9ATDP1PKM
SCHEMBL11659631 0.87 PPARA (0.48) KMT2AMEN1RAB9ATDP1PKM
SCHEMBL11037929 0.86 SIRT2 (0.55) KMT2AMEN1RAB9ATDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 74 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4401459-A POTENTIATION OF AN N-METHOXYUREA BY A 2-/PHENYL- OR PYRIDYLOXYPHENYLOXY-/ACETATE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1983-08-30 US claimed
EP-0003835-B1 A HYDROXY-UREA, PROCESS FOR PRODUCING THE SAME AND A PROCESS FOR PRODUCING A PHENYL-SUBSTITUTED N-METHOXY-N-METHYL-UREA SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1983-03-02 EP claimed
US-4349379-A N'-(4-(4-METHYL-PHENETHYLOXY)PHENYL)-N-METHOXY-N-METHYLUREA AND PHENOLIC SOLVENT SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1982-09-14 US claimed
US-4283222-A HERBICIDE, EMULSIFIER, SOLVENTS AND SURFACTANTS SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1981-08-11 US claimed
US-4263219-A METHYLATION IN TWO-PHASE REACTION MEDIUM SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1981-04-21 US claimed
JP-59106405-A None JP disclosed
JP-53108947-A None JP disclosed
JP-55089207-A None JP disclosed
JP-54112838-A None JP disclosed
JP-54112839-A None JP disclosed
JP-54112836-A None JP disclosed
JP-59172403-A None JP disclosed
US-4263219-A METHYLATION IN TWO-PHASE REACTION MEDIUM SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1981-04-21 US disclosed
JP-S5589207-A HERBICIDAL EMULSION COMPOSITION SUMITOMO CHEM CO LTD 1980-07-05 JP disclosed
EP-0003835-A1 A hydroxy-urea, process for producing the same and a process for producing a phenyl-substituted N-methoxy-N-methyl-urea SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1979-09-05 EP disclosed
JP-S54112839-A 4-METHYL-ALPHA(4-NITROPHENOXY)ACETOPHENONE AND ITS PREPARATION SUMITOMO CHEM CO LTD 1979-09-04 JP disclosed
JP-S54112836-A N'-4-2-(METHYLPHENYL) ETHOXY PHENYL-N-HYDROXYUREA AND ITS PREPARATION SUMITOMO CHEM CO LTD 1979-09-04 JP disclosed
JP-S54112838-A 4-2-(4-METHYLPHENYL)ETHOXYL NITROBENZENE AND ITS PREPARATION SUMITOMO CHEM CO LTD 1979-09-04 JP disclosed
US-4129436-A HERBICIDE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1978-12-12 US disclosed
JP-S53108947-A SUBSTITUTED PHENYLUREA DERIVATIVE, ITS PRODUCTION AND SELECTIVE HERBICIDE CONTAINING THE SAME SUMITOMO CHEM CO LTD 1978-09-22 JP disclosed