SCHEMBL9003246

SCHEMBL9003246

C[C@@H](C(=O)O)N(C(=O)Cc1ccccc1)c1cccc2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMPD2 O60906 1/20 0.45
TRPM8 Q7Z2W7 1/20 0.45
KMT2A Q03164 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.40
KDM4E B2RXH2 4/20 0.39
ALDH1A1 P00352 3/20 0.39
TDP1 Q9NUW8 2/20 0.39
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
TSHR P16473 2/20 0.38
HPGD P15428 2/20 0.38
MEN1 O00255 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7453131 0.87 KMT2A (0.47) SMPD2KMT2AL3MBTL1KDM4EALDH1A1
SCHEMBL7453130 0.87 KMT2A (0.47) SMPD2KMT2AL3MBTL1KDM4EALDH1A1
SCHEMBL7289060 0.84 KMT2A (0.42) SMPD2KMT2AKDM4EALDH1A1PSEN1
SCHEMBL7470147 0.82 L3MBTL1 (0.50) SMPD2KMT2AL3MBTL1KDM4EALDH1A1
SCHEMBL7443157 0.82 L3MBTL1 (0.50) SMPD2KMT2AL3MBTL1KDM4EALDH1A1
SCHEMBL2327184 0.82 HRH4 (0.40) SMPD2TRPM8KMT2AL3MBTL1KDM4E
SCHEMBL6113112 0.81 SMPD2 (0.47) SMPD2SIGMAR1AKR1B1
SCHEMBL6113113 0.81 SMPD2 (0.47) SMPD2SIGMAR1AKR1B1
SCHEMBL6119288 0.81 SMPD2 (0.47) SMPD2SIGMAR1AKR1B1
SCHEMBL7142898 0.81 SMPD2 (0.43) SMPD2KMT2AL3MBTL1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731790-A1 TACHYKININ ANTAGONISTS A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1996-09-18 EP disclosed