SCHEMBL7903407

SCHEMBL7903407

CC(C)=CCN1Cc2c(Br)ccc3[nH]c(=S)n(c23)C[C@@H]1C

nearest known ligand 0.31

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.31
DRD2 P14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7905347 0.88 HTR1A (0.32) HTR1ADRD2
Tivirapine SCHEMBL377308 0.87 HTR1A (0.31) HTR1ADRD2
SCHEMBL7908098 0.87 PARP1 (0.32) HTR1ADRD2
Tivirapine SCHEMBL3145162 0.87 HTR1A (0.31) HTR1ADRD2
SCHEMBL8844411 0.87 PARP1 (0.33) HTR1ADRD2
Tivirapine SCHEMBL8844208 0.86 HTR1A (0.31) HTR1ADRD2
SCHEMBL4062423 0.81 HTR1A (0.46) HTR1ADRD2
SCHEMBL29624058 0.81 HTR1A (0.46) HTR1ADRD2
SCHEMBL599870 0.81 HTR1A (0.46) HTR1ADRD2
Tibo SCHEMBL1077005 0.74 GRIN2D (0.31) HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5371079-A Administering to inhibit replication of HIV-1 in human cells JANSSEN PHARMACEUTICA N.V. (BE) 1994-12-06 US claimed
US-6201119-B1 2,3,4,5-TETRAHYDRO-1H-1,4-BENZODIAZEPIN-9-AMINE COMPOUNDS USEFUL AS INTERMEDIATES TO ANTIVIRALS JANSSEN PHARMACEUTICA N.V. (BE) 2001-03-13 US disclosed
US-5371079-A Administering to inhibit replication of HIV-1 in human cells JANSSEN PHARMACEUTICA N.V. (BE) 1994-12-06 US disclosed
US-5270464-A Anti-HIV-1 tetrahydroimidazo[1,4]benzodiazepin-2-(thi) ones JANSSEN PHARMACEUTICA N.V. (BE) 1993-12-14 US disclosed