Tivirapine

Tivirapine

SCHEMBL3145162

CC(C)=CCN1Cc2c(Cl)ccc3[nH]c(=S)n(c23)CC1C

nearest known ligand 0.31

Full drug profile on Sugi Atlas →

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.31
DRD2 P14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tivirapine SCHEMBL377308 1.00 HTR1A (0.31) HTR1ADRD2
Tivirapine SCHEMBL8844208 0.99 HTR1A (0.31) HTR1ADRD2
SCHEMBL7905545 0.90 HTR1A (0.32) HTR1ADRD2
SCHEMBL7905347 0.88 HTR1A (0.32) HTR1ADRD2
SCHEMBL7903407 0.87 HTR1A (0.31) HTR1ADRD2
SCHEMBL8844411 0.87 PARP1 (0.33) HTR1ADRD2
SCHEMBL8844088 0.86 HTR1A (0.32) HTR1ADRD2
SCHEMBL8844167 0.86 HTR1A (0.32) HTR1ADRD2
SCHEMBL9274799 0.85 HTR1A (0.33) HTR1ADRD2
SCHEMBL9695807 0.83 HTR1A (0.30) HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210254056-A1 IDENTIFICATION AND TARGETED MODULATION OF GENE SIGNALING NETWORKS CAMP4 THERAPEUTICS CORPORATION 2021-08-19 US disclosed
US-20190192691-A1 REGULATED BIOCIRCUIT SYSTEMS OBSIDIAN THERAPEUTICS, INC. 2019-06-27 US disclosed
EP-3146048-A2 NUCLEIC ACIDS ACTING AS DECOYS FOR THE TREATMENT OF LENTIVIRUS INFECTION INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2017-03-29 EP disclosed
WO-2015177331-A2 NUCLEIC ACIDS ACTING AS DECOYS FOR THE TREATMENT OF LENTIVIRUS INFECTION INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2015-11-26 WO disclosed
US-20100030530-A1 METHOD OF SEARCHING FOR LIGAND ASTELLAS PHARMA INC. (JP) 2010-02-04 US disclosed
EP-2065818-A1 METHOD OF SEARCHING FOR LIGAND Astellas Pharma Inc. (JP) 2009-06-03 EP disclosed