SCHEMBL7903565

SCHEMBL7903565

Cc1ccc(-c2ncn(C(=O)N3CCN(c4ccc(F)cc4)CC3)n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.48
TP53 P04637 3/20 0.47
MAPT P10636 5/20 0.47
KMT2A Q03164 3/20 0.47
LMNA P02545 3/20 0.47
MEN1 O00255 2/20 0.47
SLC6A7 Q99884 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
MAPK1 P28482 2/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
KDM4E B2RXH2 1/20 0.43
TSHR P16473 1/20 0.43
HTT P42858 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL427033 0.88 MAPK1 (0.60) AKR1C3TP53MAPTKMT2AMEN1
SCHEMBL425498 0.79 FAAH (0.58) AKR1C3MAPTKMT2ALMNAMEN1
SCHEMBL425711 0.78 AKR1C3 (0.49) AKR1C3MAPT
SCHEMBL424468 0.78 MAP4K1 (0.42) AKR1C3MAPTKMT2AMEN1
SCHEMBL27607283 0.72 AKR1C3 (0.83) AKR1C3KMT2ALMNAMEN1SLC6A7
SCHEMBL426884 0.71 PARP10 (0.56) AKR1C3TP53MAPTKMT2ALMNA
SCHEMBL15127495 0.71 MAPT (0.63) TP53MAPTKMT2ALMNAMEN1
SCHEMBL427358 0.70 DGAT1 (0.50) AKR1C3MAPTLMNAHTT
SCHEMBL426876 0.70 POLB (0.44) TP53MAPTKMT2ALMNAMEN1
SCHEMBL28483179 0.69 GFER (0.52) TP53MAPTKMT2AMEN1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010074588-A2 PHARMACEUTICAL COMPOUNDS BIAL - PORTELA & Cª, S.A. (PT) 2010-07-01 WO disclosed