SCHEMBL7904181

SCHEMBL7904181

N#Cc1c(SCc2csc(-c3ccc(Cl)cc3)n2)nc(N2CCC2)c(C#N)c1-c1ccc(CCCOC(=O)[C@@H](N)CCCN)cc1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 19/20 0.51
SLC6A3 Q01959 1/20 0.51
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HSD17B10 Q99714 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13261214 0.93 ADORA1 (0.59) ADORA1SLC6A3
SCHEMBL7895330 0.92 ADORA1 (0.59) ADORA1SLC6A3
SCHEMBL7899855 0.91 ADORA1 (0.53) ADORA1SLC6A3KDM4EMAPTHPGD
SCHEMBL7901799 0.90 ADORA1 (0.55) ADORA1SLC6A3KDM4EMAPTHPGD
SCHEMBL7901547 0.87 ADORA1 (0.48) ADORA1SLC6A3
SCHEMBL13943809 0.87 ADORA1 (0.64) ADORA1SLC6A3
SCHEMBL13227889 0.86 ADORA1 (0.54) ADORA1SLC6A3
SCHEMBL13227902 0.85 ADORA1 (0.54) ADORA1SLC6A3
SCHEMBL13261219 0.85 ADORA1 (0.53) ADORA1SLC6A3
SCHEMBL7902944 0.84 ADORA1 (0.53) ADORA1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2391620-B1 ALKYLAMINE-SUBSTITUTED DICYANOPYRIDINE AND AMINO ACID ESTER PRODRUGS THEREOF BAYER IP GMBH (DE) 2014-05-07 EP disclosed
WO-2010086101-A1 ALKYLAMINE-SUBSTITUTED DICYANOPYRIDINE AND AMINO ACID ESTER PRODRUGS THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-08-05 WO disclosed