SCHEMBL7901799

SCHEMBL7901799

N#Cc1c(SCc2csc(-c3ccc(Cl)cc3)n2)nc(N2CCC2)c(C#N)c1-c1ccc(CCCOC(=O)CCN)cc1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 19/20 0.55
SLC6A3 Q01959 1/20 0.55
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13260960 0.92 ADORA1 (0.63) ADORA1SLC6A3
SCHEMBL7895333 0.91 ADORA1 (0.63) ADORA1SLC6A3
SCHEMBL7904181 0.90 ADORA1 (0.51) ADORA1SLC6A3KDM4EMAPTHPGD
SCHEMBL7901547 0.89 ADORA1 (0.48) ADORA1SLC6A3
SCHEMBL7899855 0.89 ADORA1 (0.53) ADORA1SLC6A3KDM4EMAPTHPGD
Trifluoroacetic Acid SCHEMBL3726381 0.88 ADORA1 (0.58) ADORA1SLC6A3
Trifluoroacetic Acid SCHEMBL3728377 0.87 ADORA1 (0.58) ADORA1SLC6A3
SCHEMBL7900548 0.87 ADORA1 (0.55) ADORA1SLC6A3KDM4E
SCHEMBL13227890 0.85 ADORA1 (0.58) ADORA1SLC6A3
SCHEMBL21134572 0.85 ADORA1 (0.65) ADORA1SLC6A3KDM4EMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010086101-A1 ALKYLAMINE-SUBSTITUTED DICYANOPYRIDINE AND AMINO ACID ESTER PRODRUGS THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-08-05 WO disclosed